MetaADEDB 2.0 @ LMMD
Drug resistance
(UMLS:C0013203)
Definition:
Diminished or failed response of an organism, disease or tissue to the intended effectiveness of a chemical or drug. It should be differentiated from DRUG TOLERANCE which is the progressive diminution of the susceptibility of a human or animal to the effects of a drug, as a result of continued administration.
UMLS ID:
C0013203
MeSH ID:
D004351
Classification:
Name:
Physiological Phenomena
MeSH Tree Number(s):
G07.690.773.984
Synonym(s)
1.
Drug resistance
2.
Drug Resistance
3.
Drug Resistance Process
4.
Drug resistance, NOS
5.
Refractory drug response
6.
drug resistance
7.
drug-related disorder resistance
8.
drugs resistance
9.
resistance drug
Associated Drug(s)
NameNumber of ReportsReference(s)Data Source
1Imatinib MesylateFAERS: 256
Canada Vigilance: 16
Canada Vigilance
US FAERS
2Imatinib MesylateFAERS: 163
Canada Vigilance: 7
Canada Vigilance
OFFSIDES
US FAERS
3NevirapineFAERS: 151OFFSIDES
US FAERS
4LamivudineFAERS: 112OFFSIDES
US FAERS
5GefitinibFAERS: 90US FAERS
6Erlotinib HydrochlorideFAERS: 81US FAERS
7LinezolidFAERS: 77OFFSIDES
US FAERS
8entecavirFAERS: 62US FAERS
9CiprofloxacinFAERS: 49US FAERS
104-methyl-N-(3-(4-methylimidazol-1-yl)-5-(trifluoromethyl)phenyl)-3-((4-pyridin-3-ylpyrimidin-2-yl)amino)benzamideFAERS: 40
Canada Vigilance: 7
Canada Vigilance
US FAERS
11osimertinibFAERS: 37US FAERS
12LevofloxacinFAERS: 35US FAERS
13VoriconazoleFAERS: 32OFFSIDES
US FAERS
14ClopidogrelFAERS: 27US FAERS
15efavirenzFAERS: 27OFFSIDES
US FAERS
16ClozapineFAERS: 25
Canada Vigilance: 4
Canada Vigilance
US FAERS
17AcyclovirFAERS: 24US FAERS
18GanciclovirFAERS: 24
Canada Vigilance: 1
Canada Vigilance
OFFSIDES
US FAERS
19dolutegravirFAERS: 24
Canada Vigilance: 2
Canada Vigilance
US FAERS
20Erlotinib HydrochlorideFAERS: 23US FAERS
21FluconazoleFAERS: 23US FAERS
22ItraconazoleFAERS: 23US FAERS
23AfatinibFAERS: 21US FAERS
24DasatinibFAERS: 20
Canada Vigilance: 1
Canada Vigilance
US FAERS
25OseltamivirFAERS: 20
Canada Vigilance: 2
Canada Vigilance
US FAERS
26DaptomycinFAERS: 19
Canada Vigilance: 15
Canada Vigilance
US FAERS
27WarfarinFAERS: 19US FAERS
28fexofenadineFAERS: 18US FAERS
29TenofovirFAERS: 17
Canada Vigilance: 5
Canada Vigilance
OFFSIDES
US FAERS
30TenofovirFAERS: 16
Canada Vigilance: 5
Canada Vigilance
OFFSIDES
US FAERS
31adefovir dipivoxilFAERS: 16
Canada Vigilance: 1
Canada Vigilance
OFFSIDES
US FAERS
32CyclosporineFAERS: 15OFFSIDES
US FAERS
33MethotrexateFAERS: 15US FAERS
34OseltamivirFAERS: 15OFFSIDES
US FAERS
35Atazanavir SulfateFAERS: 14US FAERS
36CabergolineFAERS: 14OFFSIDES
US FAERS
37LenalidomideFAERS: 14US FAERS
38MeropenemFAERS: 14US FAERS
39ValacyclovirFAERS: 14
Canada Vigilance: 2
Canada Vigilance
US FAERS
40ceftolozane, tazobactam drug combinationFAERS: 14US FAERS
41ledipasvir, sofosbuvir drug combinationFAERS: 13
Canada Vigilance: 1
Canada Vigilance
US FAERS
42LopinavirFAERS: 12
Canada Vigilance: 1
Canada Vigilance
OFFSIDES
US FAERS
43PCI 32765FAERS: 12US FAERS
44TelbivudineFAERS: 12US FAERS
45VancomycinFAERS: 12US FAERS
46BortezomibFAERS: 11US FAERS
47CaspofunginFAERS: 11US FAERS
48MeloxicamFAERS: 11US FAERS
49PrednisoloneFAERS: 11US FAERS
50TriumeqFAERS: 11US FAERS
51AlendronateFAERS: 10US FAERS
52CeftriaxoneFAERS: 10US FAERS
53ClindamycinFAERS: 10US FAERS
54Elvitegravir, Cobicistat, Emtricitabine, Tenofovir Disoproxil Fumarate Drug CombinationFAERS: 10
Canada Vigilance: 2
Canada Vigilance
US FAERS
55LetrozoleFAERS: 10US FAERS
56MaravirocFAERS: 10US FAERS
57MicafunginFAERS: 10OFFSIDES
US FAERS
58OlanzapineFAERS: 10US FAERS
59benzoylecgonineFAERS: 10US FAERS
60Abiraterone AcetateFAERS: 9
Canada Vigilance: 1
Canada Vigilance
US FAERS
61ColchicineFAERS: 9US FAERS
62MetronidazoleFAERS: 9US FAERS
63RivaroxabanFAERS: 9US FAERS
64SorafenibFAERS: 9OFFSIDES
US FAERS
65ValganciclovirFAERS: 9US FAERS
66ceritinibFAERS: 9US FAERS
67ponatinibFAERS: 9US FAERS
68EnfuvirtideFAERS: 8US FAERS
69ImipenemFAERS: 8US FAERS
70RifampinFAERS: 8OFFSIDES
US FAERS
71VemurafenibFAERS: 8US FAERS
72avibactam, ceftazidime drug combinationFAERS: 8US FAERS
73ColistinFAERS: 7OFFSIDES
US FAERS
74HhAntag691FAERS: 7US FAERS
75MDV 3100FAERS: 7
Canada Vigilance: 1
Canada Vigilance
US FAERS
76TemozolomideFAERS: 7US FAERS
77TigecyclineFAERS: 7US FAERS
78ValganciclovirFAERS: 7US FAERS
79acalabrutinibFAERS: 7US FAERS
80olaparibFAERS: 7US FAERS
812-[(E)-[1-(2-Amino-1,3-thiazol-4-yl)-2-[[(2S,3S)-2-methyl-4-oxo-1-sulfoazetidin-3-yl]amino]-2-oxoethylidene]amino]oxy-2-methylpropanoic acid;(2S)-2,6-diaminohexanoic acidFAERS: 6
Canada Vigilance: 1
Canada Vigilance
US FAERS
82ClopidogrelFAERS: 6OFFSIDES
US FAERS
83DocetaxelFAERS: 6US FAERS
84LevetiracetamFAERS: 6OFFSIDES
US FAERS
85LoratadineFAERS: 6US FAERS
86Ruxolitinib phosphateFAERS: 6US FAERS
87AmoxicillinFAERS: 5US FAERS
88AzithromycinFAERS: 5US FAERS
89ClarithromycinFAERS: 5OFFSIDES
US FAERS
90DaptomycinFAERS: 5US FAERS
91EtoposideFAERS: 5US FAERS
92Lopinavir/RitonavirFAERS: 5
Canada Vigilance: 1
Canada Vigilance
US FAERS
93MetforminFAERS: 5US FAERS
94OctreotideFAERS: 5US FAERS
95OctreotideFAERS: 5
Canada Vigilance: 1
Canada Vigilance
US FAERS
96PregabalinFAERS: 5US FAERS
97Valproic AcidFAERS: 5US FAERS
98AnastrozoleFAERS: 4US FAERS
99AripiprazoleFAERS: 4US FAERS
100BaclofenFAERS: 4US FAERS
101DarunavirFAERS: 4OFFSIDES
US FAERS
102DexamethasoneFAERS: 4US FAERS
103Emtricitabine, Rilpivirine, Tenofovir Drug CombinationFAERS: 4US FAERS
104ErtapenemFAERS: 4US FAERS
105IbuprofenFAERS: 4US FAERS
106NaproxenFAERS: 4US FAERS
107NuvaRingFAERS: 4OFFSIDES
US FAERS
108Quetiapine FumarateFAERS: 4US FAERS
109Raltegravir PotassiumFAERS: 4
Canada Vigilance: 2
Canada Vigilance
US FAERS
110RifaximinFAERS: 4US FAERS
111SertralineFAERS: 4US FAERS
112ThyroxineFAERS: 4US FAERS
113TobramycinFAERS: 4US FAERS
114ZidovudineFAERS: 4OFFSIDES
US FAERS
115bivalirudinFAERS: 4US FAERS
116carfilzomibFAERS: 4US FAERS
117AIC246FAERS: 3US FAERS
118Amoxicillin-Potassium Clavulanate CombinationFAERS: 3US FAERS
119AmpicillinFAERS: 3OFFSIDES
US FAERS
120AspirinFAERS: 3US FAERS
121CetirizineFAERS: 3US FAERS
122CiprofloxacinFAERS: 3US FAERS
123DoripenemFAERS: 3US FAERS
124FluticasoneFAERS: 3US FAERS
125GabapentinFAERS: 3US FAERS
126JulucaFAERS: 3US FAERS
127LapatinibFAERS: 3US FAERS
128MidazolamFAERS: 3US FAERS
129MirtazapineFAERS: 3US FAERS
130OfloxacinFAERS: 3US FAERS
131Prasugrel HydrochlorideFAERS: 3US FAERS
132PrednisoneFAERS: 3
Canada Vigilance: 3
Canada Vigilance
US FAERS
133RibavirinFAERS: 3US FAERS
134RisperidoneFAERS: 3US FAERS
135RivastigmineFAERS: 3US FAERS
136SertralineFAERS: 3US FAERS
137Sildenafil CitrateFAERS: 3US FAERS
138TerbinafineFAERS: 3US FAERS
139TicagrelorFAERS: 3US FAERS
140TolvaptanFAERS: 3US FAERS
141VoseviFAERS: 3US FAERS
142WarfarinFAERS: 3US FAERS
143abacavir, lamivudine drug combinationFAERS: 3US FAERS
144apremilastFAERS: 3US FAERS
145cefprozilFAERS: 3US FAERS
146elbasvir-grazoprevir drug combinationFAERS: 3US FAERS
147gemcitabineFAERS: 3US FAERS
148pazopanibFAERS: 3US FAERS
149pimecrolimusFAERS: 3OFFSIDES
US FAERS
150posaconazoleFAERS: 3OFFSIDES
US FAERS
151ziprasidoneFAERS: 3US FAERS
1524-hydroxybutyric acidFAERS: 2US FAERS
153AcetaminophenFAERS: 2US FAERS
154AlbuterolFAERS: 2US FAERS
155AzathioprineFAERS: 2US FAERS
156BromocriptineFAERS: 2US FAERS
157BuprenorphineFAERS: 2US FAERS
158CeftriaxoneFAERS: 2US FAERS
159CefuroximeFAERS: 2US FAERS
160Cilastatin, Imipenem Drug CombinationFAERS: 2US FAERS
161CinacalcetFAERS: 2US FAERS
162DoxorubicinFAERS: 2US FAERS
163DoxycyclineFAERS: 2US FAERS
164DoxycyclineFAERS: 2US FAERS
165ErythromycinFAERS: 2
Canada Vigilance: 1
Canada Vigilance
OFFSIDES
US FAERS
166EverolimusFAERS: 2US FAERS
167Fingolimod HydrochlorideFAERS: 2US FAERS
168FluorouracilFAERS: 2US FAERS
169FluoxetineFAERS: 2US FAERS
170FoscarnetFAERS: 2US FAERS
171FulvestrantFAERS: 2
Canada Vigilance: 1
Canada Vigilance
US FAERS
172FurosemideFAERS: 2US FAERS
173GanciclovirFAERS: 2US FAERS
174GentamicinsFAERS: 2US FAERS
175Glatiramer AcetateFAERS: 2US FAERS
176IsoniazidFAERS: 2US FAERS
177LamotrigineFAERS: 2US FAERS
178LidodermFAERS: 2US FAERS
179LiraglutideFAERS: 2US FAERS
180MethotrexateFAERS: 2US FAERS
181MethylphenidateFAERS: 2US FAERS
182MethylprednisoloneFAERS: 2
Canada Vigilance: 1
Canada Vigilance
US FAERS
183MiconazoleFAERS: 2US FAERS
184MorphineFAERS: 2OFFSIDES
US FAERS
185OxcarbazepineFAERS: 2US FAERS
186PaclitaxelFAERS: 2US FAERS
187PanobinostatFAERS: 2US FAERS
188PropranololFAERS: 2US FAERS
189QuinidineFAERS: 2US FAERS
190Rosuvastatin CalciumFAERS: 2US FAERS
191SimeprevirFAERS: 2US FAERS
192SirolimusFAERS: 2US FAERS
193SumatriptanFAERS: 2US FAERS
194SunitinibFAERS: 2US FAERS
195TopiramateFAERS: 2US FAERS
196ValacyclovirFAERS: 2US FAERS
197Venlafaxine HydrochlorideFAERS: 2US FAERS
198Viekira PakFAERS: 2US FAERS
199Zoledronic AcidFAERS: 2
Canada Vigilance: 1
Canada Vigilance
US FAERS
200brexpiprazoleFAERS: 2US FAERS
201cefuroxime axetilFAERS: 2US FAERS
202cisatracuriumFAERS: 2US FAERS
203emtricitabine tenofovir alafenamideFAERS: 2US FAERS
204pazopanibFAERS: 2US FAERS
205pomalidomideFAERS: 2US FAERS
206AcetylcysteineFAERS: 1US FAERS
207AlprazolamFAERS: 1US FAERS
208AmlodipineFAERS: 1US FAERS
209AmoxicillinFAERS: 1US FAERS
210ArthrotecFAERS: 1US FAERS
211AtorvastatinFAERS: 1US FAERS
212AtovaquoneFAERS: 1US FAERS
213Atropine sulphateFAERS: 1US FAERS
214AxitinibFAERS: 1US FAERS
215Bendamustine HydrochlorideFAERS: 1US FAERS
216BosentanFAERS: 1US FAERS
217BromocriptineFAERS: 1US FAERS
218BudesonideFAERS: 1US FAERS
219BupropionFAERS: 1US FAERS
220CapecitabineFAERS: 1US FAERS
221CarbamazepineFAERS: 1US FAERS
222Carbidopa, levodopa, and entacaponeFAERS: 1US FAERS
223CarnitineFAERS: 1US FAERS
224CefdinirFAERS: 1US FAERS
225CefepimeFAERS: 1US FAERS
226CelecoxibFAERS: 1US FAERS
227CidofovirFAERS: 1OFFSIDES
US FAERS
228CitalopramFAERS: 1US FAERS
229ClindamycinFAERS: 1US FAERS
230ClobazamFAERS: 1
Canada Vigilance: 1
Canada Vigilance
US FAERS
231DeferasiroxFAERS: 1US FAERS
232DiazepamFAERS: 1US FAERS
233DiclofenacFAERS: 1US FAERS
234Dimethyl FumarateFAERS: 1US FAERS
235Emtricitabine, Tenofovir Disoproxil Fumarate Drug CombinationFAERS: 1US FAERS
236EsomeprazoleFAERS: 1US FAERS
237EvotazFAERS: 1US FAERS
238FentanylFAERS: 1US FAERS
239Fexofenadine hydrochloride and pseudoephedrine hydrochlorideFAERS: 1US FAERS
240FidaxomicinFAERS: 1US FAERS
241FinasterideFAERS: 1US FAERS
242FluoxetineFAERS: 1
Canada Vigilance: 1
Canada Vigilance
US FAERS
243GS-7340FAERS: 1US FAERS
244GoserelinFAERS: 1US FAERS
245HaloperidolFAERS: 1US FAERS
246HomoharringtonineFAERS: 1US FAERS
247HydrochlorothiazideFAERS: 1US FAERS
248HydroxyureaFAERS: 1OFFSIDES
US FAERS
249HydroxyzineFAERS: 1US FAERS
250ImiquimodFAERS: 1US FAERS
251IndomethacinFAERS: 1US FAERS
252Insulin GlargineFAERS: 1US FAERS
253InsulinFAERS: 1US FAERS
254IrbesartanFAERS: 1US FAERS
255IrinotecanFAERS: 1US FAERS
256IsotretinoinFAERS: 1US FAERS
257IvermectinFAERS: 1US FAERS
258Lisdexamfetamine DimesylateFAERS: 1US FAERS
259LoperamideFAERS: 1US FAERS
260Loratadine and pseudoephedrine sulfateFAERS: 1US FAERS
261LosartanFAERS: 1US FAERS
262MercaptopurineFAERS: 1US FAERS
263MesalamineFAERS: 1US FAERS
264MetforminFAERS: 1US FAERS
265MethylergonovineFAERS: 1US FAERS
266MethylphenidateFAERS: 1US FAERS
267Methylprednisolone HemisuccinateFAERS: 1US FAERS
268MitoxantroneFAERS: 1US FAERS
269ModafinilFAERS: 1US FAERS
270Mometasone FuroateFAERS: 1US FAERS
271MoxifloxacinFAERS: 1US FAERS
272MupirocinFAERS: 1US FAERS
273Mycophenolic AcidFAERS: 1US FAERS
274NaltrexoneFAERS: 1US FAERS
275NitrofurantoinFAERS: 1
Canada Vigilance: 1
Canada Vigilance
US FAERS
276Olmesartan MedoxomilFAERS: 1US FAERS
277OmeprazoleFAERS: 1US FAERS
278OrlistatFAERS: 1US FAERS
279OxacillinFAERS: 1US FAERS
280Paliperidone PalmitateFAERS: 1US FAERS
281PantoprazoleFAERS: 1US FAERS
282PenicillamineFAERS: 1US FAERS
283Penicillin GFAERS: 1OFFSIDES
US FAERS
284PhenytoinFAERS: 1OFFSIDES
US FAERS
285PrezcobixFAERS: 1US FAERS
286PrimaquineFAERS: 1US FAERS
287PropofolFAERS: 1US FAERS
288PropranololFAERS: 1US FAERS
289QVA149FAERS: 1US FAERS
290Quetiapine FumarateFAERS: 1US FAERS
291Raltegravir PotassiumFAERS: 1US FAERS
292RamiprilFAERS: 1US FAERS
293RilpivirineFAERS: 1US FAERS
294RitonavirFAERS: 1US FAERS
295RocuroniumFAERS: 1US FAERS
296SaquinavirFAERS: 1OFFSIDES
US FAERS
297SevofluraneFAERS: 1US FAERS
298Sitagliptin PhosphateFAERS: 1US FAERS
299Solifenacin SuccinateFAERS: 1US FAERS
300StavudineFAERS: 1OFFSIDES
US FAERS
301TacrolimusFAERS: 1
Canada Vigilance: 1
Canada Vigilance
US FAERS
302TamoxifenFAERS: 1
Canada Vigilance: 1
Canada Vigilance
US FAERS
303TerbinafineFAERS: 1US FAERS
304TetrabenazineFAERS: 1US FAERS
305TetracyclineFAERS: 1US FAERS
306ThalidomideFAERS: 1US FAERS
307TiclopidineFAERS: 1US FAERS
308TinzaparinFAERS: 1US FAERS
309TrazodoneFAERS: 1US FAERS
310Triamcinolone AcetonideFAERS: 1US FAERS
311TriamcinoloneFAERS: 1US FAERS
312TriiodothyronineFAERS: 1US FAERS
313Ursodeoxycholic AcidFAERS: 1US FAERS
314ValsartanFAERS: 1US FAERS
315VancomycinFAERS: 1
Canada Vigilance: 2
Canada Vigilance
US FAERS
316VyxeosFAERS: 1US FAERS
317argatrobanFAERS: 1OFFSIDES
US FAERS
318atovaquone, proguanil drug combinationFAERS: 1US FAERS
319benazeprilFAERS: 1US FAERS
320bosutinibFAERS: 1US FAERS
321carbidopa, levodopa drug combinationFAERS: 1US FAERS
322carbidopa, levodopa drug combinationFAERS: 1US FAERS
323clindamycin phosphateFAERS: 1US FAERS
324dabrafenibFAERS: 1US FAERS
325darifenacinFAERS: 1US FAERS
326ecallantideFAERS: 1US FAERS
327edoxabanFAERS: 1US FAERS
328eltrombopagFAERS: 1US FAERS
329etravirineFAERS: 1US FAERS
330fanasil, pyrimethamine drug combinationFAERS: 1US FAERS
331gemcitabineFAERS: 1US FAERS
332idelalisibFAERS: 1US FAERS
333insulin glulisineFAERS: 1US FAERS
334isavuconazoleFAERS: 1US FAERS
335isavuconazoleFAERS: 1US FAERS
336lamivudine, zidovudine drug combinationFAERS: 1US FAERS
337levocetirizineFAERS: 1US FAERS
338linaclotideFAERS: 1US FAERS
339midostaurinFAERS: 1US FAERS
340mirabegronFAERS: 1US FAERS
341montelukastFAERS: 1US FAERS
342niraparibFAERS: 1US FAERS
343palbociclibFAERS: 1US FAERS
344quinupristin-dalfopristinFAERS: 1US FAERS
345regorafenibFAERS: 1US FAERS
346reviparinFAERS: 1US FAERS
347suvorexantFAERS: 1US FAERS
348tofacitinibFAERS: 1US FAERS
349trametinibFAERS: 1US FAERS
350treprostinilFAERS: 1US FAERS
351venetoclaxFAERS: 1US FAERS
352zolmitriptanFAERS: 1US FAERS
353AcitretinOFFSIDES
354AmikacinCanada Vigilance: 1Canada Vigilance
OFFSIDES
355BezafibrateOFFSIDES
356CaspofunginOFFSIDES
357CaspofunginOFFSIDES
358CefotaximeOFFSIDES
359CortisoneOFFSIDES
360Cyproterone AcetateOFFSIDES
361CytarabineOFFSIDES
362DapsoneOFFSIDES
363DidanosineOFFSIDES
364ErtapenemOFFSIDES
365EstradiolOFFSIDES
366EthambutolOFFSIDES
367FlucytosineOFFSIDES
368FoscarnetOFFSIDES
369GliclazideOFFSIDES
370IndinavirOFFSIDES
371LevodopaOFFSIDES
372MeclizineOFFSIDES
373MethimazoleOFFSIDES
374MicafunginCanada Vigilance: 1Canada Vigilance
375NafronylOFFSIDES
376NelfinavirOFFSIDES
377NeostigmineOFFSIDES
378NorepinephrineOFFSIDES
379Paliperidone PalmitateCanada Vigilance: 1Canada Vigilance
380PamidronateOFFSIDES
381Penicillin VOFFSIDES
382SulfadiazineOFFSIDES
383SumatriptanOFFSIDES
384TaurineOFFSIDES
385ThiopentalOFFSIDES
386TrifluoperazineOFFSIDES
387VareniclineCanada Vigilance: 1Canada Vigilance
388VigabatrinOFFSIDES
389VincristineOFFSIDES
390VindesineOFFSIDES
391VirginiamycinOFFSIDES
392ZalcitabineOFFSIDES
393abacavirOFFSIDES
394amprenavirOFFSIDES
395calcium acetateOFFSIDES
396desloratadineCanada Vigilance: 1Canada Vigilance
397entacaponeOFFSIDES
398eprosartanOFFSIDES
399fosamprenavirOFFSIDES
400isepamicinOFFSIDES
401liposomal amphotericin BOFFSIDES
402liposomal doxorubicinCanada Vigilance: 1Canada Vigilance
403polaprezincOFFSIDES
404prednisolone acetateOFFSIDES
405tipranavirOFFSIDES
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