2025

5
2025 6th. Month
ERRα-Predictor: A Framework of Ensemble Models for Prediction of ERRα Binders, Antagonists, and Agonists Using Artificial Intelligence
Authors: Le Xiong, Jiahao Xu, Hongbo Yu, Weihua Li, Xinmin Li, Wenxiang Song, Jingwei Zhang, Yun Tang*, Guixia Liu*
Journal: Journal of Chemical Information and Modeling
Information 2025 | 65(13) | 6809–6822
2025 6th. Month
In Silico Prediction of pKa Values Using Explainable Deep Learning Methods
Authors: Chen Yang, Changda Gong, Zhixing Zhang, Jiaojiao Fang, Weihua Li, Guixia Liu, Yun Tang
Journal: Journal of Pharmaceutical Analysis
Information 2025 | 15(6) | 101174
2025 4th. Month
TCnet: a novel strategy to predict target combination of Alzheimer’s disease via network-based methods
Authors: Yue CY, Chen BY, Pan F, Wang Z, Yu HB, Liu GX, Li WH, Wang R*, Tang Y*
Journal: Journal of Chemical Information and Modeling
Information 2025
2025 3th. Month
Cocry-pred: a dynamic resource propagation method for cocrystal prediction
Authors: Song WX#, Peng R#, Yu HB, Zhan ML, Liu GX, Li WH, Ren GB, Zhu B*, Tang Y*
Journal: Journal of Chemical Information and Modeling
Information 2025 | 65(6) | 2868-2881
2025 3th. Month
Fluor-Predictor: An Interpretable Tool for Multiproperty Prediction and Retrieval of Fluorescent Dyes
Authors: Wenxiang Song, Le Xiong, Xinmin Li, Yuyang Zhang, Binya Wang, Guixia Liu, Weihua Li, Youjun Yang*, Yun Tang*
Journal: Journal of Chemical Information and Modeling
Information 2025 | 65(6) | 2868–2881

2024

4
2024 11th. Month
ToxGIN: an In silico prediction model for peptide toxicity via graph isomorphism networks integrating peptide sequence and structure information
Authors: Qiule Yu, Zhixing Zhang, Guixia Liu, Weihua Li, Yun Tang*
Journal: Briefings in Bioinformatics
Information 2024 | 25(6) | bbae583
2024 10th. Month
In Silico Prediction of ERRα Agonists Based on Combined Features and Stacking Ensemble Method
Authors: Jiahao Xu, Zejun Huang, Hao Duan, Weihua Li, Jingyan Zhuang, Le Xiong, Yun Tang, Guixia Liu
Journal: ChemMedChem
Information 2024 | 19(20) | e202400298
2024 6th. Month
人工智能在抗癌肽研发中的应用与挑战
Authors: Zhixing Zhang, Hua Deng, Yun Tang
Journal: 中国药科大学学报
Information 2024 | Vol.55(3) | 347 − 356
2024 3th. Month
MedChatZH: A tuning LLM for traditional Chinese medicine consultations
Authors: Yang Tan, Zhixing Zhang, Mingchen Li, Fei Pan, Hao Duan, Zijie Huang, Hua Deng, Zhuohang Yu, Chen Yang, Guoyang Shen, Peng Qi, Chengyuan Yue, Yuxian Liu, Liang Hong, Huiqun Yu, Guisheng Fan, Yun Tang
Journal: Computers in Biology and Medicine
Information 2024 | Vol.172 | 108290

2022

16
2022 12th. Month
Development of In Silico Models for Predicting Potential Time-Dependent Inhibitors of Cytochrome P450 3A4
Authors: Minjie Xu, Zhou Lu, Zengrui Wu, Minyan Gui, Guixia Liu, Yun Tang*, Weihua Li*
Journal: Molecular Pharmaceutics
Information 2022 | 20(1) | 194–205
2022 11th. Month
In silico prediction of chemical aquatic toxicity by multiple machine learning and deep learning approaches
Authors: Minjie Xu, Hongbin Yang, Guixia Liu, Yun Tang, Weihua Li*
Journal: Journal of Applied Toxicology
Information 2022 | 42(11) | 1766-1776
2022 10th. Month
In silico prediction of potential drug-induced nephrotoxicity with machine learning methods
Authors: Yuning Gong, Dan Teng, Yimeng Wang, Yaxin Gu, Zengrui Wu, Weihua Li, Yun Tang*, Guixia Liu*
Journal: Journal of Applied Toxicology
Information 2022 | 42(10) | 1639-1650
2022 9th. Month
In Silico Prediction of Human and Rat Liver Microsomal Stability via Machine Learning Methods
Authors: Longqiang Li, Zhou Lu, Guixia Liu, Yun Tang, Weihua Li*
Journal: Chemical Research in Toxicology
Information 2022 | 35(9) | 1614–1624
2022 9th. Month
Profiling prediction of nuclear receptor modulators with multi-task deep learning methods: toward the virtual screening
Authors: Jiye Wang, Chaofeng Lou, Guixia Liu, Weihua Li, Zengrui Wu, Yun Tang*
Journal: Briefings in Bioinformatics
Information 2022 | 23(5) | bbac351
2022 9th. Month
Drug Repurposing for Newly Emerged Diseases via Network-based Inference on a Gene-disease-drug Network
Authors: Li Qin, Jiye Wang, Zengrui Wu, Weihua Li, Guixia Liu, Yun Tang*
Journal: Molecular Informatics
Information 2022 | 41(9) | e2200001
2022 8th. Month
Prediction of anti-inflammatory peptides by a sequence-based stacking ensemble model named AIPStack
Authors: Hua Deng, Chaofeng Lou, Zengrui Wu, Weihua Li, Guixia Liu, Yun Tang*
Journal: iScience
Information 2022 | 25(9) | 104967
2022 7th. Month
Mechanistic Studies on the Stereoselectivity of FFAR1 Modulators
Authors: Dan Teng, Yang Zhou, Yun Tang, Guixia Liu*, Yaoquan Tu*
Journal: Journal of Chemical Information and Modeling
Information 2022 | 61(15) | 3664–3675
2022 7th. Month
In silico prediction of UGT-mediated metabolism in drug-like molecules via graph neural network
Authors: Mengting Huang, Chaofeng Lou, Zengrui Wu, Weihua Li, Philip W. Lee, Yun Tang*, Guixia Liu*
Journal: Journal of Cheminformatics
Information 2022
2022 6th. Month
Investigation of the mechanism of Shen Qi Wan prescription in the treatment of T2DM via network pharmacology and molecular docking
Authors: Piaopiao Zhao, Xiaoxiao Zhang, Yuning Gong, Weihua Li, Zengrui Wu, Yun Tang*, Guixia Liu*
Journal: in Silico Pharmacology
Information 2022 | 10(9)
2022 5th. Month
IDL-PPBopt: A Strategy for Prediction and Optimization of Human Plasma Protein Binding of Compounds via an Interpretable Deep Learning Method
Authors: Chaofeng Lou, Hongbin Yang, Jiye Wang, Mengting Huang, Weihua Li, Guixia Liu, Philip W. Lee, Yun Tang*
Journal: Journal of Chemical Information and Modeling
Information 2022 | 62(11) | 2788–2799
2022 3th. Month
A multitask GNN-based interpretable model for discovery of selective JAK inhibitors
Authors: Yimeng Wang, Yaxin Gu, Chaofeng Lou, Yuning Gong, Zengrui Wu, Weihua Li, Yun Tang*, Guixia Liu*
Journal: Journal of Cheminformatics
Information 2022 | 14(1) | 16
2022 3th. Month
ADENet: a novel network-based inference method for prediction of drug adverse events
Authors: Zhuohang Yu, Zengrui Wu*, Weihua Li, Guixia Liu, Yun Tang*
Journal: Briefings in Bioinformatics
Information 2022 | 23(2) | bbab580
2022 2th. Month
In Silico Prediction of Potential Drug Combinations for Type 2 Diabetes Mellitus by an Integrated Network and Transcriptome Analysis
Authors: Dan Teng, Yuning Gong, Zengrui Wu, Weihua Li, Yun Tang*, Guixia Liu*
Journal: Chemmedchem
Information 2022 | 17(3) | e202100620
2022 1th. Month
wSDTNBI: a novel network-based inference method for virtual screening
Authors: Zengrui Wu#, Hui Ma#, Zehui Liu#, Lulu Zheng, Zhuohang Yu, Shuying Cao, Wenqing Fang, Lili Wu, Weihua Li, Guixia Liu, Jin Huang, Yun Tang*
Journal: Chemical Science
Information 2022 | 13(4) | 1060-1079
2022 1th. Month
Discovery of New Estrogen-Related Receptor α Agonists via a Combination Strategy Based on Shape Screening and Ensemble Docking
Authors: Dongping Li, Kexin Jiang, Dan Teng, Zengrui Wu, Weihua Li, Yun Tang*, Rui Wang*, Guixia Liu*
Journal: Journal of Chemical Information and Modeling
Information 2022 | 62(3) | 486–497

2021

9
2021
Insights into the Molecular Mechanisms of Liuwei Dihuang Decoction via Network Pharmacology
Authors: Jianhui Chen, Dan Teng, Zengrui Wu, Weihua Li, Yuqian Feng, Yun Tang*, Guixia Liu*
Journal: Chem. Res. Toxicol.
Information 2021 | 34(1) | 91-102
2021
In silico prediction of chemical acute contact toxicity on honey bees via machine learning methods
Authors: Xuan Xu, Piaopiao Zhao, Zhiyuan Wang, Xiaoxiao Zhang, Zengrui Wu, Weihua Li, Yun Tang*, Guixia Liu*
Journal: Toxicol. In Vitro
Information 2021 | Vol.72 | 105089
2021
In silico prediction of mitochondrial toxicity of chemicals using machine learning methods
Authors: Piaopiao Zhao, Yayuan Peng, Xuan Xu, Zhiyuan Wang, Zengrui Wu, Weihua Li, Yun Tang*, Guixia Liu*
Journal: J. Appl. Toxicol.
Information 2021 | Vol.DOI | 10
2021
In silico prediction of chemical respiratory toxicity via machine learning
Authors: Zhiyuan Wang, Piaopiao Zhao, Xiaoxiao Zhang, Xuan Xu, Weihua Li, Guixia Liu, Yun Tang*
Journal: Comput. Toxicol.
Information 2021 | Vol.18 | 100155
2021
Assessment of CYP2C9 Structural Models for Site of Metabolism Prediction
Authors: Xiaoxiao Zhang, Minjie Xu, Zengrui Wu, Guixia Liu, Yun Tang, Weihua Li*
Journal: ChemMedChem
Information 2021 | Vol.DOI | 10
2021
Twin drug design, synthesis and evaluation of diosgenin derivatives as multitargeted agents for the treatment of vascular dementia
Authors: Guixiang Yang, Jiamin Sun, Lulu Zheng, Li Zhang, Jie Li, Haixian Gan, Yan Huang, Jin Huang, Xingxing Diao, Yun Tang*, Rui Wang*, Lei Ma*
Journal: Bioorg. Med. Chem.
Information 2021 | Vol.37 | 116109
2021
Homotropic Cooperativity of Midazolam Metabolism by Cytochrome P450 3A4: Insight from Computational Studies
Authors: Junhao Li, Yue Chen, Yun Tang, Weihua Li*, Yaoquan Tu*
Journal: J. Chem. Inf. Model.
Information 2021 | 61(5) | 2418-2426
2021
Pathway-Based Drug Repurposing with DPNetinfer: A Method to Predict Drug–Pathway Associations via Network-Based Approaches
Authors: Jiye Wang, Zengrui Wu, Yayuan Peng, Weihua Li, Guixia Liu, Yun Tang*
Journal: J. Chem. Inf. Model.
Information 2021 | 61(5) | 2475-2485
2021
Discovery of Natural Products Targeting NQO1 via an Approach Combining Network-Based Inference and Identification of Privileged Substructures
Authors: Zengrui Wu, Qiaohui Wang, Hongbin Yang, Jiye Wang, Weihua Li, Guixia Liu, Yi Yang, Yuzheng Zhao*, Yun Tang*
Journal: J. Chem. Inf. Model.
Information 2021 | 61(5) | 2486-2498

2020

14
2020
In Silico Prediction of Human Renal Clearance of Compounds Using Quantitative Structure-Pharmacokinetic Relationship Models
Authors: Jianhui Chen, Hongbin Yang, Lan Zhu, Zengrui Wu, Weihua Li, Yun Tang*, Guixia Liu*
Journal: Chem. Res. Toxicol.
Information 2020 | 33(2) | 640-650
2020
Mechanistic Insights into the Regio- and Stereoselectivities of Testosterone and Dihydrotestosterone Hydroxylation Catalyzed by CYP3A4 and CYP19A1
Authors: Junhao Li, Yun Tang, Weihua Li*, Yaoquan Tu*
Journal: Chem. - Eur. J.
Information 2020 | 26(28) | 6214-6223
2020
Computational Approaches to Identify Structural Alerts and Their Applications in Environmental Toxicology and Drug Discovery
Authors: Hongbin Yang, Chaofeng Lou, Weihua Li, Guixia Liu, Yun Tang*
Journal: Chem. Res. Toxicol.
Information 2020 | 33(6) | 1312-1322
2020
Computational Insight into the Allosteric Activation Mechanism of Farnesoid X Receptor
Authors: Yue Chen, Junhao Li, Zengrui Wu, Guixia Liu, Honglin Li, Yun Tang*, Weihua Li*
Journal: J. Chem. Inf. Model.
Information 2020 | 60(3) | 1540-1550
2020
In Silico Prediction of Metabolic Epoxidation for Drug-like Molecules via Machine Learning Methods
Authors: Jiajing Hu, Yingchun Cai, Weihua Li, Guixia Liu, Yun Tang*
Journal: Mol. Inf.
Information 2020 | 39(8) | 1900178
2020
In silico prediction of binding capacity and interaction forces of organic compounds with α- and β-cyclodextrins
Authors: Peiwen Di, Jianhui Chen, Liping Liu, Weihua Li, Yun Tang*, Guixia Liu*
Journal: J. Mol. Liq.
Information 2020 | Vol.302 | 112585
2020
Drug repositioning by prediction of drug's anatomical therapeutic chemical code via network-based inference approaches
Authors: Yayuan Peng, Manjiong Wang, Yixiang Xu, Zengrui Wu, Jiye Wang, Chao Zhang, Guixia Liu, Weihua Li, Jian Li*, Yun Tang*
Journal: Briefings Bioinf.
Information 2020 | 22(2) | 2058–2072
2020
Computational Insights into Molecular Activation and Positive Cooperative Mechanisms of FFAR1 Modulators
Authors: Dan Teng, Jianhui Chen, Dongping Li, Zengrui Wu, Weihua Li, Yun Tang*, Guixia Liu*
Journal: J. Chem. Inf. Model.
Information 2020 | 60(6) | 3214-3230
2020
In silico prediction of chemical neurotoxicity using machine learning
Authors: Changsheng Jiang, Piaopiao Zhao, Weihua Li, Yun Tang*, Guixia Liu*
Journal: Toxicol. Res.
Information 2020 | 9(3) | 164–172
2020
NetInfer: A Web Server for Prediction of Targets and Therapeutic and Adverse Effects via Network-Based Inference Methods
Authors: Zengrui Wu, Yayuan Peng, Zhuohang Yu, Weihua Li, Guixia Liu, Yun Tang*
Journal: J. Chem. Inf. Model.
Information 2020 | 60(8) | 3687-3691
2020
Dissecting the Structural Plasticity and Dynamics of Cytochrome P450 2B4 by Molecular Dynamics Simulations
Authors: Junhao Li, Yang Zhou, Yun Tang, Weihua Li*, Yaoquan Tu*
Journal: J. Chem. Inf. Model.
Information 2020 | 60(10) | 5026-5035
2020
Strategy for Efficient Discovery of Cocrystals via a Network-Based Recommendation Model
Authors: Lulu Zheng, Bin Zhu, Zengrui Wu, Xiaoxue Fang, Minghuang Hong, Guixia Liu, Weihua Li, Guobin Ren*, Yun Tang*
Journal: Cryst. Growth Des.
Information 2020 | 20(10) | 6820-6830
2020
Insights into the mechanism of Arnebia euchroma on leukemia via network pharmacology approach
Authors: Biting Wang, Zengrui Wu*, Jiye Wang, Weihua Li, Guixia Liu, Bo Zhang, Yun Tang*
Journal: BMC Complementary Med. Ther.
Information 2020 | 20(1) | 322
2020
MetaADEDB 2
Authors: Zhuohang Yu, Zengrui Wu*, Weihua Li, Guixia Liu, Yun Tang*
Journal: 0: a comprehensive database on adverse drug events. Bioinformatics
Information 2020 | Vol.DOI | 10

2019

13
2019
Computational Prediction of Site of Metabolism for UGT-Catalyzed Reactions
Authors: Yingchun Cai, Hongbin Yang, Weihua Li, Guixia Liu, Philip W Lee, Yun Tang*
Journal: J. Chem. Inf. Model.
Information 2019 | 59(3) | 1085-1095
2019
Computational insights into the different catalytic activities of CYP3A4 and CYP3A5 toward schisantherin E
Authors: Yuhan Xue, Junhao Li, Zengrui Wu, Guixia Liu, Yun Tang, Weihua Li*
Journal: Chem. Biol. Drug Des.
Information 2019 | 93(5) | 854–864
2019
In silico prediction of chemical reproductive toxicity using machine learning
Authors: Changsheng Jiang, Hongbin Yang, Peiwen Di, Weihua Li, Yun Tang*, Guixia Liu*
Journal: J. Appl. Toxicol.
Information 2019 | 39(6) | 844-854
2019
Computational insights into the interaction mechanisms of estrogen-related receptor alpha with endogenous ligand cholesterol
Authors: Dongping Li, Yingchun Cai, Dan Teng, Weihua Li, Yun Tang*, Guixia Liu*
Journal: Chem. Biol. Drug Des.
Information 2019 | 94(1) | 1316-1329
2019
In Silico Prediction of Endocrine Disrupting Chemicals Using Single-Label and Multilabel Models
Authors: Lixia Sun, Hongbin Yang, Yingchun Cai, Weihua Li, Guixia Liu, Yun Tang*
Journal: J. Chem. Inf. Model.
Information 2019 | 59(3) | 973-982
2019
Insights into the antineoplastic mechanism of Chelidonium majus via systems pharmacology approach
Authors: Xinzhe Xiao, Zehui Chen, Zengrui Wu, Tianduanyi Wang, Weihua Li, Guixia Liu, Bo Zhang*, Yun Tang*
Journal: Quant. Biol.
Information 2019 | 7(1) | 42-53
2019
Prediction of the skin sensitising potential and potency of compounds via mechanism-based binary and ternary classification models
Authors: Peiwen Di, Yongmin Yin, Changsheng Jiang, Yingchun Cai, Weihua Li, Yun Tang*, Guixia Liu*
Journal: Toxicol. In Vitro
Information 2019 | Vol.59 | 204-214
2019
Insights into mechanisms and severity of drug-induced liver injury via computational systems toxicology approach
Authors: Yayuan Peng, Zengrui Wu*, Hongbin Yang, Yingchun Cai, Guixia Liu, Weihua Li, Yun Tang*
Journal: Toxicol. Lett.
Information 2019 | Vol.312 | 22-33
2019
A novel derivative of artemisinin inhibits cell proliferation and metastasis via down-regulation of cathepsin K in breast cancer
Authors: Xiangyu Gu, Yayuan Peng, Yuyu Zhao, Xin Liang*, Yun Tang*, Jianwen Liu*
Journal: Eur. J. Pharmacol.
Information 2019 | Vol.858 | 172382
2019
Design, synthesis and biological evaluation of chalcones as reversers of P-glycoprotein-mediated multidrug resistance
Authors: Huanhuan Yin, Jingjing Dong, Yingchun Cai, Ximeng Shi, Hao Wang, Guixia Liu, Yun Tang*, Jianwen Liu*, Lei Ma*
Journal: Eur. J. Med. Chem.
Information 2019 | Vol.180 | 350-366
2019
Prediction of the allergic mechanism of haptens via a reaction-substructure-compound-target-pathway network system
Authors: Peiwen Di, Zengrui Wu, Hongbin Yang, Weihua Li, Yun Tang*, Guixia Liu*
Journal: Toxicol. Lett.
Information 2019 | Vol.317 | 68-81
2019
Insights into the interaction mechanisms of estrogen-related receptor alpha (ERRα) with ligands via molecular dynamics simulations
Authors: Dongping Li, Yingchun Cai, Dan Teng, Zengrui Wu, Weihua Li, Yun Tang*, Guixia Liu*
Journal: J. Biomol. Struct. Dyn.
Information 2019 | 38(13) | 3867-3878
2019
Design, synthesis and evaluation of diosgenin carbamate derivatives as multitarget anti-Alzheimer's disease agents
Authors: Guixiang Yang, Yan Huang, Lulu Zheng, Li Zhang, Lin Su, Yuhang Wu, Jie Li, Licheng Zhou, Jin Huang, Yun Tang*, Rui Wang*, Lei Ma*
Journal: Eur. J. Med. Chem.
Information 2019 | Vol.187 | 111913

2018

14
2018
In Silico Prediction of Chemical Toxicity for Drug Design Using Machine Learning Methods and Structural Alerts
Authors: Hongbin Yang, Lixia Sun, Weihua Li, Guixia Liu, Yun Tang*
Journal: Front. Chem.
Information 2018 | Vol.6 | 30
2018
Corrigendum: In Silico Prediction of Chemical Toxicity for Drug Design Using Machine Learning Methods and Structural Alerts
Authors: Hongbin Yang, Lixia Sun, Weihua Li, Guixia Liu, Yun Tang*
Journal: Front. Chem.
Information 2018 | Vol.6 | 129
2018
Lee, Yun Tang*
Authors: Yingchun Cai, Hongbin Yang, Weihua Li, Guixia Liu, Philip W
Journal: Multiclassification Prediction of Enzymatic Reactions for Oxidoreductases and Hydrolases Using Reaction Fingerprints and Machine Learning Methods. J. Chem. Inf. Model.
Information 2018 | 58(6) | 1169-1181
2018
A Computational Systems Pharmacology Approach to Investigate Molecular Mechanisms of Herbal Formula Tian-Ma-Gou-Teng-Yin for Treatment of Alzheimer's Disease
Authors: Tianduanyi Wang, Zengrui Wu, Lixia Sun, Weihua Li, Guixia Liu, Yun Tang*
Journal: Front. Chem.
Information 2018 | Vol.9 | 668
2018
Identification of Nontoxic Substructures: A New Strategy to Avoid Potential Toxicity Risk
Authors: Hongbin Yang, Lixia Sun, Weihua Li, Guixia Liu, Yun Tang*
Journal: Toxicol. Sci.
Information 2018 | 165(2) | 396–407
2018
In silico estimation of chemical aquatic toxicity on crustaceans using chemical category methods
Authors: Qianqian Cao, Lin Liu, Hongbin Yang, Yingchun Cai, Weihua Li, Guixia Liu, Philip W Lee, Yun Tang*
Journal: Environ. Sci.: Processes Impacts
Information 2018 | 20(9) | 1234-1243
2018
In Silico Prediction of Blood–Brain Barrier Permeability of Compounds by Machine Learning and Resampling Methods
Authors: Zhuang Wang, Hongbin Yang, Zengrui Wu, Tianduanyi Wang, Weihua Li, Yun Tang*, Guixia Liu*
Journal: ChemMedChem.
Information 2018 | 13(20) | 2189–2201
2018
admetSAR 2
Authors: Hongbin Yang, Chaofeng Lou, Lixia Sun, Jie Li, Yingchun Cai, Zhuang Wang, Weihua Li, Guixia Liu, Yun Tang*
Journal: 0: web-service for prediction and optimization of chemical ADMET properties. Bioinformatics.
Information 2018 | 35(6) | 1067-1069
2018
Computational Insight Into Vitamin K1 ω-Hydroxylation by Cytochrome P450 4F2
Authors: Junhao Li, Hongxiao Zhang, Guixia Liu, Yun Tang, Yaoquan Tu*, Weihua Li*
Journal: Front. Pharmacol.
Information 2018 | Vol.9 | 1065
2018
ADMETopt: A Web Server for ADMET Optimization in Drug Design via Scaffold Hopping
Authors: Hongbin Yang, Lixia Sun, Zhuang Wang, Weihua Li, Guixia Liu, Yun Tang*
Journal: J. Chem. Inf. Model.
Information 2018 | 58(10) | 2051-2056
2018
Network-Based Methods for Prediction of Drug-Target Interactions
Authors: Zengrui Wu, Weihua Li, Guixia Liu, Yun Tang*
Journal: Front. Pharmacol.
Information 2018 | Vol.9 | 1134
2018
Prediction of Farnesoid X Receptor Disruptors with Machine Learning Methods
Authors: Yue Chen, Hongbin Yang, Zengrui Wu, Guixia Liu, Yun Tang, Weihua Li*
Journal: Chem. Res. Toxicol.
Information 2018 | 31(11) | 1128-1137
2018
ADMET-score – a comprehensive scoring function for evaluation of chemical drug-likeness
Authors: Longfei Guan, Hongbin Yang, Yingchun Cai, Lixia Sun, Peiwen Di, Weihua Li, Guixia Liu, Yun Tang*
Journal: MedChemComm.
Information 2018 | 10(1) | 148-157
2018
Modified rivaroxaban microparticles for solid state properties improvement based on drug-protein/polymer supramolecular interactions
Authors: Ning Chen, Peiwen Di, Shangqi Ning, Wenjun Jiang, Qiufang Jing, Guobin Ren, Yan Liu, Yun Tang, Zhongyu Xu, Guixia Liu*, Fuzheng Ren*
Journal: Powder Technol.
Information 2018 | Vol.344 | 819–829

2017

14
2017
Computational Investigation of Ligand Binding to the Peripheral Site in CYP3A4: Conformational Dynamics and Inhibitor Discovery
Authors: Hanwen Du, Junhao Li, Yingchun Cai, Hongxiao Zhang, Guixia Liu, Yun Tang*, Weihua Li*
Journal: J. Chem. Inf. Model.
Information 2017 | 57(3) | 616-626
2017
Insights into the molecular mechanisms of Polygonum multiflorum Thunb-induced liver injury: a computational systems toxicology approach
Authors: Yinyin Wang, Jie Li, Zengrui Wu, Bo Zhang, Hongbin Yang, Qin Wang, Yingchun Cai, Guixia Liu, Weihua Li, Yun Tang*
Journal: Acta Pharmacol. Sin.
Information 2017 | 38(5) | 719-732
2017
In Silico Prediction of Chemicals Binding to Aromatase with Machine Learning Methods
Authors: Hanwen Du, Yingchun Cai, Hongbin Yang, Hongxiao Zhang, Yuhan Xue, Guixia Liu, Yun Tang, Weihua Li*
Journal: Chem. Res. Toxicol.
Information 2017 | 30(5) | 1209-1218
2017
Improving the physicochemical properties of bicalutamide by complex formation with bovine serum albumin
Authors: Congbin Yang, Peiwen Di, Jinping Fu, Hui Xiong, Qiufang Jing, Guobin Ren, Yun Tang, Wenyun Zheng, Guixia Liu*, Fuzheng Ren*
Journal: Eur. J. Pharm. Sci.
Information 2017 | Vol.106 | 381-392
2017
Evaluation of Different Methods for Identification of Structural Alerts Using Chemical Ames Mutagenicity Data Set as a Benchmark
Authors: Hongbin Yang, Jie Li, Zengrui Wu, Weihua Li, Guixia Liu, Yun Tang*
Journal: Chem. Res. Toxicol.
Information 2017 | 30(6) | 1355-1364
2017
In silico prediction of chemical subcellular localization via multi-classification methods
Authors: Hongbin Yang, Xiao Li, Yingchun Cai, Qin Wang, Weihua Li, Guixia Liu, Yun Tang*
Journal: MedChemComm.
Information 2017 | 8(6) | 1225-1234
2017
In silico prediction of pesticide aquatic toxicity with chemical category approaches
Authors: Fuxing Li, Defang Fan, Hao Wang, Hongbin Yang, Weihua Li, Yun Tang*, Guixia Liu*
Journal: Toxicol. Res.
Information 2017 | 6(6) | 831–842
2017
Quantitative and Systems Pharmacology
Authors: Jiansong Fang, Zengrui Wu, Chuipu Cai, Qi Wang, Yun Tang*, Feixiong Cheng*
Journal: 1. In Silico Prediction of Drug–Target Interactions of Natural Products Enables New Targeted Cancer Therapy. J. Chem. Inf. Model.
Information 2017 | 57(11) | 2657-2671
2017
In Silico Prediction of Compounds Binding to Human Plasma Proteins by QSAR Models
Authors: Lixia Sun, Hongbin Yang, Jie Li, Tianduanyi Wang, Weihua Li, Guixia Liu, Yun Tang*
Journal: ChemMedChem.
Information 2017 | 13(6) | 572–581
2017
Computational insights into the subtype selectivity and “message-address-efficacy” mechanisms of opioid receptors through JDTic binding and unbinding
Authors: Jianxin Cheng, Tao Cheng, Weihua Li, Guixia Liu, Weiliang Zhu, Yun Tang*
Journal: Acta Pharmacol. Sin.
Information 2017 | 39(3) | 482-491
2017
Quantitative and systems pharmacology 2
Authors: Zengrui Wu, Weiqiang Lu, Weiwei Yu, Tianduanyi Wang, Weihua Li, Guixia Liu, Hankun Zhang, Xiufeng Pang, Jin Huang, Mingyao Liu*, Feixiong Cheng*, Yun Tang*
Journal: In silico polypharmacology of G protein-coupled receptor ligands via network-based approaches. Pharmacol. Res.
Information 2017 | Vol.129 | 400-413
2017
Computational insights into the G-protein-biased activation and inactivation mechanisms of the μ opioid receptor
Authors: Jianxin Cheng, Tao Cheng, Weihua Li, Guixia Liu, Weiliang Zhu, Yun Tang*
Journal: Acta Pharmacol. Sin.
Information 2017 | 39(1) | 154-164
2017
Network pharmacological mechanisms of Vernonia anthelmintica (L
Authors: Jiye Wang, Hong Chen, Yinyin Wang, Xiaoqin Wang, Hanying Chen, Mei Zhang, Yun Tang*, Bo Zhang*
Journal: ) in the treatment of vitiligo: Isorhamnetin induction of melanogenesis via up-regulation of melanin-biosynthetic genes. BMC Syst. Biol.
Information 2017 | 11(1) | 103
2017
In silico prediction of chemical genotoxicity using machine learning methods and structural alerts
Authors: Defang Fan, Hongbin Yang, Fuxing Li, Lixia Sun, Peiwen Di, Weihua Li, Yun Tang*, Guixia Liu*
Journal: Toxicol. Res.
Information 2017 | 7(2) | 211-220

2016

9
2016
Effects of protein flexibility and active site water molecules on the prediction of sites of metabolism for cytochrome P450 2C19 substrates
Authors: Junhao Li, Jinya Cai, Haixia Su, Hanwen Du, Juan Zhang, Shihui Ding, Guixia Liu, Yun Tang*, Weihua Li*
Journal: Mol. BioSyst.
Information 2016 | 12(3) | 868-878
2016
Lee, Yun Tang*
Authors: Chen Zhang, Yuan Zhou, Shikai Gu, Zengrui Wu, Wenjie Wu, Changming Liu, Kaidong Wang, Guixia Liu, Weihua Li, Philip W
Journal: In silico prediction of hERG potassium channel blockage by chemical category approaches. Toxicol. Res.
Information 2016 | 5(2) | 570-582
2016
Computational insight into conformational states of glucagon-like peptide-1 receptor (GLP-1R) and its binding mode with GLP-1
Authors: Juan Zhang, Shikai Gu, Xianqiang Sun, Weihua Li, Yun Tang*, Guixia Liu*
Journal: RSC Adv.
Information 2016 | 6(16) | 13490-13497
2016
Computational insights into different inhibition modes of the κ-opioid receptor with antagonists LY2456302 and JDTic
Authors: Jianxin Cheng, Weihua Li, Guixia Liu, Weiliang Zhu, Yun Tang*
Journal: RSC Adv.
Information 2016 | 6(17) | 13626-13635
2016
SDTNBI: an integrated network and chemoinformatics tool for systematic prediction of drug–target interactions and drug repositioning
Authors: Zengrui Wu, Feixiong Cheng, Jie Li, Weihua Li, Guixia Liu, Yun Tang*
Journal: Brief Bioinform.
Information 2016 | Vol.DOI | 10
2016
Interactions of omeprazole-based analogues with cytochrome P450 2C19: a computational study
Authors: Junhao Li, Hanwen Du, Zengrui Wu, Haixia Su, Guixia Liu, Yun Tang*, Weihua Li*
Journal: Mol. BioSyst.
Information 2016 | 12(6) | 1913-1921
2016
Network-based identification of microRNAs as potential pharmacogenomic biomarkers for anticancer drugs
Authors: Jie Li, Kecheng Lei, Zengrui Wu, Weihua Li, Guixia Liu, Jianwen Liu, Feixiong Cheng, Yun Tang*
Journal: Oncotarget
Information 2016 | 7(29) | 45584-45596
2016
In silico prediction of chemical mechanism of action via an improved network-based inference method
Authors: Zengrui Wu, Weiqiang Lu, Dang Wu, Anqi Luo, Hanping Bian, Jie Li, Weihua Li, Guixia Liu, Jin Huang*, Feixiong Cheng, Yun Tang*
Journal: Br. J. Pharmacol.
Information 2016 | 173(23) | 3372-3385
2016
Computational investigation of the interaction mechanism between the estrogen related receptor α and its agonists
Authors: Fuxing Li, Xianqiang Sun, Yingchun Cai, Defang Fan, Weihua Li, Yun Tang*, Guixia Liu*
Journal: RSC Adv.
Information 2016 | 6(96) | 94119-94127

2015

10
2015
Lee*, Yun Tang*
Authors: Chen Zhang, Feixiong Cheng, Lu Sun, Shulin Zhuang, Weihua Li, Guixia Liu, Philip W
Journal: In silico prediction of chemical toxicity on avian species using chemical category approaches. Chemosphere
Information 2015 | Vol.122 | 280-287
2015
Discovery of New Non-Steroidal Farnesoid X Receptor Modulators Through 3D Shape Similarity Search and Structure-Based Virtual Screening
Authors: Lei Wang, Pei Si, Yayun Sheng, Yingjie Chen, Ping Wan, Xu Shen, Yun Tang, Lili Chen*, Weihua Li*
Journal: Chem. Biol. Drug Des.
Information 2015 | Vol.85 | 481-487
2015
Lee, Yun Tang*
Authors: Lu Sun, Chen Zhang, Yingjie Chen, Xiao Li, Shulin Zhuang, Weihua Li, Guixia Liu, Philip W
Journal: In silico prediction of chemical aquatic toxicity with chemical category approaches and substructural alerts. Toxicol. Res.
Information 2015 | Vol.4 | 452-463
2015
FXR antagonism of NSAIDs contributes to drug-induced liver injury identified by systems pharmacology approach
Authors: Weiqiang Lu, Feixiong Cheng, Jing Jiang, Chen Zhang, Xiaokang Deng, Zhongyu Xu, Shien Zou*, Xu Shen, Yun Tang*, Jin Huang*
Journal: Scientific Reports
Information 2015 | Vol.5 | 8114
2015
Residues remote from the binding pocket control the antagonist selectivity towards the corticotropin-releasing factor receptor-1
Authors: Xianqiang Sun, Jianxin Cheng, Xu Wang, Yun Tang*, Hans Agren, Yaoquan Tu*
Journal: Scientific Reports
Information 2015 | Vol.5 | 8066
2015
In Silico Estimation of Chemical Carcinogenicity with Binary and Ternary Classification Methods
Authors: Xiao Li, Zheng Du, Jie Wang, Zengrui Wu, Weihua Li, Guixia Liu, Xu Shen, Yun Tang*
Journal: Mol. Inform.
Information 2015 | Vol.34 | 228-235
2015
Quantitative Regression Models for the Prediction of Chemical Properties by an Efficient Workflow
Authors: Yongmin Yin, Congying Xu, Shikai Gu, Weihua Li, Guixia Liu*, Yun Tang*
Journal: Mol. Inform.
Information 2015 | 34(10) | 679-688
2015
Association between cigarette smoking and Parkinson's disease: A meta-analysis
Authors: Xiao Li, Weihua Li, Guixia Liu, Xu Shen, Yun Tang*
Journal: Arch. Gerontol. Geriat.
Information 2015 | 61(3) | 510-516
2015
Mendrick, Yun Tang*, Feixiong Cheng*
Authors: Chen Zhang, Huixiao Hong, Donna L
Journal: Biomarker-based drug safety assessment in the age of systems pharmacology: from foundational to regulatory science. Biomark. Med.
Information 2015 | 9(11) | 1241-1252
2015
Computational insights into inhibitory mechanism of azole compounds against human aromatase
Authors: Jinya Cai, Junhao Li, Juan Zhang, Shihui Ding, Guixia Liu, Weihua Li*, Yun Tang*
Journal: RSC Adv.
Information 2015 | 5(110) | 90871-90880

2014

6
2014
Computational prediction of microRNA networks incorporating environmental toxicity and disease etiology
Authors: Jie Li, Zengrui Wu, Feixiong Cheng, Weihua Li, Guixia Liu, Yun Tang*
Journal: Scientific Reports
Information 2014 | Vol.4 | 5576
2014
Selective ligands of estrogen receptor β discovered using pharmacophore mapping and structure-based virtual screening
Authors: Lei Chen, Dang Wu, Hanping Bian, Guanglin Kuang, Jing Jiang, Weihua Li, Guixia Liu, Shien Zou*, Jin Huang, Yun Tang*
Journal: Acta Pharmacol. Sin.
Information 2014 | Vol.35 | 1333-1341
2014
Structure-based ensemble-QSAR model: a novel approach to the study of the EGFR tyrosine kinase and its inhibitors
Authors: Xianqiang Sun, Lei Chen, Yaozong Li, Weihua Li, Guixia Liu, Yaoquan Tu*, Yun Tang*
Journal: Acta Pharmacol. Sin.
Information 2014 | Vol.35 | 301-310
2014
In Silico Prediction of Chemical Acute Oral Toxicity Using Multi-Classification Methods
Authors: Xiao Li, Lei Chen, Feixiong Cheng, Zengrui Wu, Hanping Bian, Congying Xu, Weihua Li, Guixia Liu, Xu Shen, Yun Tang*
Journal: J. Chem. Inf. Model.
Information 2014 | 54(4) | 1061-1069
2014
Effects of protein flexibility on the site of metabolism prediction for CYP2A6 substrates
Authors: Yayun Sheng, Yingjie Chen, Lei Wang, Guixia Liu, Weihua Li*, Yun Tang*
Journal: J. Mol. Graph. Model.
Information 2014 | Vol.54 | 90-99
2014
Computational models to predict endocrine-disrupting chemical binding with androgen or oestrogen receptors
Authors: Yingjie Chen, Feixiong Cheng, Lu Sun, Weihua Li, Guixia Liu, Yun Tang*
Journal: Ecotox. Environ. Safe.
Information 2014 | Vol.110 | 280-287

2013

8
2013
In Silico ADMET Prediction: Recent Advances, Current Challenges and Future Trends
Authors: Feixiong Cheng, Weihua Li, Guixia Liu, Yun Tang*
Journal: Curr Top Med Chem
Information 2013 | 13(11) | 1273-1289
2013
Adverse Drug Events: Database Construction and In Silico Prediction
Authors: Feixiong Cheng, Weihua Li, Xichuan Wang, Yadi Zhou, Zengrui Wu, Jie Shen and Yun Tang
Journal: J. Chem. Inf. Model.
Information 2013 | 53(4) | 744-752
2013
Lee, Yun Tang*
Authors: Feixiong Cheng, Weihua Li, Yadi Zhou, Jie Li, Jie Shen, Philip W
Journal: Prediction of Human Genes and Diseases Targeted by Xenobiotics Using Predictive Toxicogenomics-Derived Models (PTDMs). Mol. BioSyst
Information 2013 | 9(6) | 1316-1325
2013
Prediction of Polypharmacological Profiles of Drugs by the Integration of Chemical, Side Effects and Therapeutic Space
Authors: Feixiong Cheng, Weihua Li, Zengrui Wu, Xichuan Wang, Chen Zhang, Jie Li, Guixia Liu and Yun Tang
Journal: J. Chem. Inf. Model.
Information 2013 | 53(4) | 753-762
2013
The role of benzoic acid in proline-catalyzed asymmetric michael addition: A density functional theory study
Authors: Hongwei Shi, Xiangui Huang, Guixia Liu*, Kunqian Yu, Congying Xu, Weihua Li, Bubing Zeng*, Yun Tang*
Journal: Int. J. Quantum. Chem.
Information 2013 | 113(9) | 1339-1348
2013
Catalytic Mechanism of Cytochrome P450 2D6 for 4-Hydroxylation of Aripiprazole: A QM/MM Study
Authors: Rongwei Shi, Weihua Li, Guixia Liu, Yun Tang*
Journal: Chinese J. Chem.
Information 2013 | 31(9) | 1219-1227
2013
Design, synthesis and biological evaluation of organophosphorous-homodimers as dual binding site acetylcholinesterase inhibitors
Authors: Ruliang Xie, Qianfei Zhao, Tao Zhang, Jing Fang , Xiangdong Mei, Jun Ning*, Yun Tang*
Journal: Bioorg. Med. Chem.
Information 2013 | 21(1) | 278-282
2013
Computational insights into the binding modes of Sr-Rex with cofactor NADH/NAD+ and operator DNA
Authors: Yanyan Chu, Weihua Li, Jianfeng Wang, Guixia Liu, Yun Tang*
Journal: J. Mol. Model.
Information 2013 | 19(8) | 3143-3151

2012

19
2012
Novel triazolyl bis-amino acid derivatives readily synthesized via click chemistry as potential corrosion inhibitors for mild steel in HCl
Authors: Qiong Deng, Hong-Wei Shi, Bao-Qin Chen, Xiao-Peng He, Guixia Liu, Yun Tang, Yi-Tao Long, Guo-Rong Chen
Journal: Corros. Sci.
Information 2012 | Vol.57 | 220-227
2012
In Silico Investigation of Interactions between Human Cannabinoid Receptor-1 and Its Antagonists
Authors: Guanglin Kuang, Guoping Hu, Xianqiang Sun, Weihua Li, Guixia Liu, Yun Tang*
Journal: J. Mol. Model.
Information 2012 | 18(8) | 3831-3845
2012
Lee* and Yun Tang*
Authors: Feixiong Cheng, Yutaka Ikenaga, Yadi Zhou, Yue Yu, Weihua Li, Jie Shen, Zheng Du, Lei Chen, Congyin Xu, Guixia Liu, Philip W
Journal: In Silico Assessment of Chemical Biodegradability. J. Chem. Inf. Model.
Information 2012 | 52(3) | 655-669
2012
Investigation of indazole unbinding pathways in CYP2E1 by molecular dynamics simulations
Authors: Zhonghua Shen, Feixiong Cheng, You Xu, Jing Fu, Wen Xiao, Jie Shen, Guixia Liu, Weihua Li*, and Yun Tang*
Journal: PLoS One
Information 2012 | 7(3) | e33500
2012
Synthesis and biological evaluation of quinazoline and quinoline bearing 2,2,6,6-tetramethylpiperidine-N-oxyl as potential epidermal growth factor receptor (EGFR) tyrosine kinase inhibitors and EPR bio-probe agents
Authors: Siyuan Li, Chunying Guo, Xianqiang Sun, Yaozong Li, Hongli Zhao, Dongmei Zhan, Minbo Lan*, Yun Tang*
Journal: Euro. J. Med. Chem.
Information 2012 | Vol.49 | 271-278
2012
Prediction of Drug-Target Interactions and Drug Repositioning via Network-Based Inference
Authors: Feixiong Cheng, Chuang Liu, Jing Jiang, Weiqiang Lu, Weihua Li, Guixia Liu, Weixing Zhou, Jin Huang, and Yun Tang*
Journal: PLoS Comput Biol
Information 2012 | 8(5) | e1002503
2012
Discovery of novel EGFR tyrosine kinase inhibitors by structure-based virtual screening
Authors: Siyuan Li, Xianqiang Sun, Hongli Zhao, Yun Tang*, Minbo Lan*
Journal: Bioorg. Med. Chem. Lett.
Information 2012 | 22(12) | 4004-4009
2012
Discovery and Structure-Activity Analysis of Selective Estrogen Receptor Modulators via Similarity-Based Virtual Screening
Authors: Jie Shen, Jing Jiang, Guanglin Kuang, Chengfang Tan, Guixia Liu, Jin Huang*, and Yun Tang*
Journal: Euro. J. Med. Chem.
Information 2012 | Vol.54 | 188-196
2012
Performance Evaluation of 2D Fingerprint and 3D Shape Similarity Methods in Virtual Screening
Authors: Guoping Hu, Guanglin Kuang, Wen Xiao, Weihua Li, Guixia Liu, Yun Tang*
Journal: J. Chem. Inf. Model
Information 2012 | 52(5) | 1103-1113
2012
Prediction of Chemical-Protein Interactions: Multitarget-QSAR versus Computational Chemogenomic Methods
Authors: Feixiong Cheng, Yadi Zhou, Jie Li, Weihua Li, Guixia Liu and Yun Tang*
Journal: Mol. BioSyst.
Information 2012 | Vol.8 | 2373-2384
2012
Identification of diverse dipeptidyl peptidase IV inhibitors via structure-based virtual screening
Authors: Cui Li, Weiqiang Lu, Chunhua Lu, Wen Xiao,Xu Shen, Jin Huang, Guixia Liu*, Yun Tang*
Journal: J. Mol. Model.
Information 2012 | Vol.18 | 4033-4042
2012
Concise CuI-Catalyzed Azide-Alkyne 1,3-Dipolar Cycloaddition Reaction Ligation Remarkably Enhances the Corrosion Inhibitive Potency of Natural Amino Acids for Mild Steel in HCl
Authors: Qiong Deng, Xiaopeng He, Hongwei Shi, Baoqin Chen, Guixia Liu, Yun Tang, Yitao Long, Guorong Chen, and Kaixian Chen
Journal: Ind. Eng. Chem. Res.
Information 2012 | Vol.51 | 7160-7169
2012
Synthesis, Structure–Activity Relationship, and Pharmacophore Modeling Studies of Pyrazole-3-Carbohydrazone Derivatives as Dipeptidyl Peptidase IV Inhibitors
Authors: Deyan Wu, Fangfang Jin, Weiqiang Lu, Jin Zhu, Cui Li, Wei Wang, Yun Tang, Hualiang Jiang, Jin Huang, Guixia Liu, and Jian Li
Journal: Chem. Biol. Drug. Des.
Information 2012 | Vol.79 | 897-906
2012
Prediction of Chemical-Protein Interactions Network with Weighted Network-based Inference Method
Authors: Feixiong Cheng, Yadi Zhou, Weihua Li, Guixia Liu and Yun Tang*
Journal: PLoS One
Information 2012 | 7(7) | e41064
2012
Lee, and Yun Tang*
Authors: Congying Xu, Feixiong Cheng, Lei Chen, Zheng Du, Weihua Li, Guixia Liu, Philip W
Journal: In Silico Prediction of Chemical Ames Mutagenicity. J. Chem. Inf. Model.
Information 2012 | 52(11) | 2840-2847
2012
Discovery of Inhibitors to Block Interactions of HIV-1 Integrase with Human LEDGF/p75 via Structure-Based Virtual Screening and Bioassays
Authors: Guoping Hu, Xi Li, Xuan Zhang, Yaozong Li, Lei Ma, Liumeng Yang, Guixia Liu, Weihua Li, Jin Huang, Xu Shen, Lihong Hu, Yongtang Zheng and Yun Tang*
Journal: J. Med. Chem.
Information 2012 | Vol.55 | 10108-10117
2012
Identification of old drugs as potential inhibitors of HIV-1 integrase-human LEDGF/p75 interaction via molecular docking
Authors: Guoping Hu, Xi Li, Xianqiang Sun, Weiqiang Lu Guixia Liu, Jin Huang, Xu Shen and Yun Tang
Journal: J. Mol. Model
Information 2012 | Vol.18 | 4995-5003
2012
Unbinding pathways of GW4064 from human farnesoid X receptor as revealed by molecular dynamics simulations
Authors: Weihua Li, Jing Fu, Feixiong Cheng, Mingyue Zheng, Jian Zhang, Guixia Liu, and Yun Tang*
Journal: J. Chem. Inf. Model.
Information 2012 | 52(11) | 3043-3052
2012
Inhibitors of HIV-1 Integrase-Human LEDGF/p75 Interaction Identified from Natural Products via Virtual Screening
Authors: Guoping Hu, Xi Li, Yaozong Li, Xianqiang Sun, Guixia Liu, Weihua Li, Jin Huang*, Xu Shen, Yun Tang
Journal: Chin. J. Chem.
Information 2012 | 30(12) | 2752-2758

2011

13
2011
Insights into binding modes of 5-HT2c receptor antagonists with ligand-based and receptor-based methods
Authors: Chunhua Lu, Fangfang Jin, Cui Li, Weihua Li, Guixia Liu*, Yun Tang*
Journal: J Mol Model
Information 2011 | 17(10) | 2513-2523
2011
Insights into subtype selectivity of opioid agonists by ligand-based and structure-based methods
Authors: Jianxin Cheng, Guixia Liu*, Jing Zhang, Zhejun Xu and Yun Tang*
Journal: J Mol Model.
Information 2011 | Vol.17 | 477-493
2011
Crucial role of the first CXXC motif of human QSOX 1b in protein thiol oxidation
Authors: Zheng Wenyun, Chu Yanyan, Yin Qin, Xu Lei, Yang Charles, Zhang Wenyao, Tang Yun*, Yang Yi*
Journal: J. Biochemistry
Information 2011 | 149(3) | 293-300
2011
Computational investigation of interactions between human H2 receptor and its agonists
Authors: Sun Xianqiang, Li Yaozong, Li Weihua, Xu Zhejun, Tang Yun*
Journal: J. Mol. Graph. Modelling
Information 2011 | 29(5) | 693-701
2011
Identification of small molecular inhibitors for Ero1p by structure-based virtual screening
Authors: Chu Yanyan, Chen Xianjun, Yang Yi*, Tang Yun*
Journal: Bioorg. Med. Chem. Lett.
Information 2011 | 21(4) | 1118-1121
2011
Lee, Tang Yun*
Authors: Cheng Feixiong, Shen Jie, Yu Yue, Li Weihua*, Liu Guixia, Philip W
Journal: In silico prediction of Tetrahymena pyriformis toxicity for diverse industrial chemicals with substructure pattern recognition and machine learning methods. Chemosphere
Information 2011 | 82(11) | 1636-1643
2011
Exploring coumarin egress channels in human cytochrome P450 2A6 by random acceleration and steered molecular dynamics simulations
Authors: Weihua Li, Jie Shen, Guixia Liu, Tang Yun*, Tyuji Hoshino*
Journal: Proteins
Information 2011 | 79(1) | 271-281
2011
Possible Ligand Release Pathway of Dipeptidyl Peptidase IV Investigated by Molecular Dynamics Simulations
Authors: Cui Li, Jie Shen, Weihua Li, Chunhua Lu, Guixia Liu*, Yun Tang*
Journal: Proteins: Structure, Function and Bioinformatics.
Information 2011 | 79(6) | 1800-1809
2011
Lee, and Yun Tang*
Authors: Feixiong Cheng, Yue Yu, Jie Shen, Lei Yang, Weihua Li*, Guixia Liu, Philip W
Journal: Classification of Cytochrome P450 Inhibitors and non-Inhibitors using Combined Classifiers. J. Chem. Inf. Model.
Information 2011 | 51(5) | 996-1011
2011
Computational insights into the different catalytic activities of CYP2A13 and CYP2A6 on NNK
Authors: You Xu, Zhonghua Shen, Jie Shen, Guixia Liu, Weihua Li*, and Yun Tang*
Journal: J. Mol. Graph. Model.
Information 2011 | Vol.30 | 1-9
2011
Computational Insights into Ligand Selectivity of Estrogen Receprors from Pharmacophore Modeling
Authors: Jing Fang, Jie Shen, Feixiong Cheng, Zhejun Xu, Guixia Liu, and Yun Tang*
Journal: Mol. Inf.
Information 2011 | Vol.30 | 539-549
2011
An Unusual (R)-Selective Epoxide Hydrolase with High Activity for Facile Preparation of Enantiopure Glycidyl Ethers
Authors: Jing Zhao, Yan-Yan Chu, Ai-Tao Li, Xin Ju, Xu-Dong Kong, Jiang Pan, Yun Tang* and Jian-He Xu*
Journal: Adv. Synth. Catal.
Information 2011 | Vol.353 | 1510-1518
2011
Click to a focused library of benzyl 6-triazolo(hydroxy)benzoic glucosides: Novel construction of PTP1B inhibitors on a sugar scaffold
Authors: Cui Li, Xiao-Peng He, Yin-Jie Zhang, Zhen Li, Li-Xin Gao, Xiao-Xin Shi, Juan Xie, Jia Li, Guo-Rong Chen*, Yun Tang*
Journal: Euro. J. Med. Chem.
Information 2011 | Vol.46 | 4212-4218

2010

6
2010
Triazole-linked benzylated glucosyl, galacotosyl and mannosyl monomers and dimmers as novel sugar scaffold-based PTP1B inhibitors
Authors: Zhang Yinjie, He Xiaopeng, Li Cui, Li Zhen, Shi Detai, Gao Lixin, Qiu Beiying, Shi Xiaoxin, Tang Yun*, Li Jia*, Chen Guorong*
Journal: Chem. Lett.
Information 2010 | 39(12) | 1261-1263
2010
Pharmacophore modeling of human adenosine receptor A2A antagonists
Authors: Zhejun Xu, Feixiong Cheng, Chenxiao Da, Guixia Liu and Yun Tang*
Journal: J. Mol .Model
Information 2010 | Vol.16 | 1867-1876
2010
Insights into binding modes of adenosine A2B antagonists with ligand-based and receptor-based methods
Authors: Feixiong Cheng, Zhejun Xu, Liu Guixia and Yun Tang*
Journal: Euro. J. Med. Chem.
Information 2010 | Vol.45 | 3459-3471
2010
Accuracy Assessment of Protein-Based Docking Programs against RNA Targets
Authors: Yaozong Li, Jie Shen, Xianqiang Sun, Weihua Li, Guixia Liu, and Yun Tang*
Journal: J. Chem. Inf. Model
Information 2010 | Vol.50 | 1134-146
2010
Estimation of ADME Properties with Substructure Pattern Recognition
Authors: Jie Shen, Feixiong Cheng, You Xu, Weihua Li,* and Yun Tang*
Journal: J. Chem. Inf. Model.
Information 2010 | Vol.50 | 1034-041
2010
Discovery of Potent Ligands for Estrogen Receptor β by Structure-Based Virtual Screening
Authors: Jie Shen, Chengfang Tan, Yanyan Zhang, Xi Li, Weihua Li, Jin Huang,,Xu Shen and Yun Tang
Journal: J. Med. Chem.
Information 2010 | Vol.53 | 5361-365

2009

4
2009
The crystal structure of a complex of acetylcholinesterase with a bis-(-)-nor-meptazinol derivative reveals disruption of the catalytic triad
Authors: Paz A, Xie Q, Greenblatt HM, Fu W, Tang Y, Silman I, Qiu ZB, Sussman JL*
Journal: J. Med. Chem.
Information 2009 | 52(8) | 2543-2549
2009
Reduced catalytic activity of P450 2A6 mutants with Coumarin: a computational investigation
Authors: Li WH, Ode H, Hoshino T*, Liu H, Tang Y*, Jiang HL
Journal: J. Chem. Theory Comput.
Information 2009 | 5(5) | 1411-1420
2009
Computational Insights into the Mechanism of Ligand Unbinding and Selectivity of Estrogen Receptors
Authors: Jie Shen, Weihua Li, Guixia Liu, Yun Tang and Hualiang Jiang
Journal: J. Phys. Chem. B
Information 2009 | 113(30) | 10436-0444
2009
Structure–function analysis of human protein Ero1-La
Authors: Yanyan Chu, Charles Yang, Xianjun Chen, Wenyun Zheng, Yi Yang* and Yun Tang,*
Journal: Biochem. Biophys. Res. Comm.
Information 2009 | Vol.389 | 645-650

2008

7
2008
Hyrtiosal, from the marine sponge Hyrtios erectus, inhibits HIV-1 integrase binding to viral DNA by a new inhibitor binding site
Authors: Du L, Shen LL, Yu ZG, Chen J, Guo YW*, Tang Y*, Shen X*, Jiang HL
Journal: ChemMedChem
Information 2008 | 3(1) | 173-180
2008
Insights into ligand selectivity in estrogen receptor isoforms: molecular dynamics simulations and binding free energy calculations
Authors: Zeng J, Li WH, Zhao YX, Liu GX*, Tang Y*, Jiang HL
Journal: J. Phys. Chem. B
Information 2008 | 112(9) | 2719-2726
2008
Probing ligand binding modes of human cytochrome P450 2J2 by homology modeling, molecular dynamics simulation, and flexible molecular docking
Authors: Li WH, Tang Y*, Liu H, Cheng JG, Zhu WL, Jiang HL
Journal: Proteins
Information 2008 | 71(2) | 938-949
2008
Insights into the interactions between HIV-1 integrase and human LEDGF/p75 by molecular dynamics simulation and free energy calculation
Authors: Zhao YX, Li WH, Zeng J, Liu GX, Tang Y*
Journal: Proteins
Information 2008 | 72(2) | 635-645
2008
In silico prediction of blood-brain partitioning using a chemometric method called genetic algorithm based variable selection
Authors: Shen J, Du YP, Zhao YX, Liu GX, Tang Y*
Journal: QSAR Comb. Sci.
Information 2008 | 27(6) | 704-717
2008
Role of acetylation and extra-cellular location of heat shock protein 90alpha in tumor cell invasion
Authors: Yang YH, Rao R, Shen J, Tang Y, Fiskus W, Nechtman J, Atadja P, Bhalla K
Journal: Cancer Res.
Information 2008 | 68(12) | 4833-4842
2008
D77, one benzoic acid derivative, functions as a novel anti-HIV-1 inhibitor targeting the interaction between integrase and cellular LEDGF/p75
Authors: Du L, Zhao YX, Chen J, Yang LM, Zheng YT, Tang Y*, Shen X*, Jiang HL
Journal: Biochem. Biophys. Res. Comm.
Information 2008 | 375(1) | 139-144

2007

2
2007
Synthesis of highly functionalized chiral cyclopentanes by catalytic enantio- and diastereoselective double Michael addition reactions
Authors: Zu L, Li H, Xie H, Wang J, Jiang W, Tang Y*, Wang W*
Journal: Angew. Chem. Int. Ed.
Information 2007 | 46(20) | 3732-3734
2007
Structure-based 3D-QSAR studies on heteroarylpiperazine derivatives as 5-HT3 receptor antagonists
Authors: Zhou YJ, Zhu LP, Tang Y*, Ye DY*
Journal: Eur. J. Med. Chem.
Information 2007 | 42(7) | 977-984

2006

4
2006
Molecular modeling and 3D-QSAR studies of indolomorphinan derivatives as kappa opioid antagonists
Authors: Li W, Tang Y*, Zheng YL, Qiu ZB*
Journal: Bioorg. Med. Chem.
Information 2006 | 14(3) | 601-610
2006
QSAR study of 4-phenylpiperidine derivatives as mu opioid agonists by neural network method
Authors: Wang XH, Tang Y*, Xie Q, Qiu ZB*
Journal: Eur. J. Med. Chem.
Information 2006 | 41(2) | 226-232
2006
Action mechanisms and structure–activity relationships of PI3Kγ inhibitors on the enzyme: a molecular modeling study
Authors: Kuang RR, Qian F, Li Z, Wei DZ*, Tang Y*
Journal: Eur. J. Med. Chem.
Information 2006 | 41(4) | 558-565
2006
New technologies of computer-aided drug design: towards target identification and new chemical entity discovery
Authors: Tang Y, Zhu WL, Chen KX, Jiang HL*
Journal: Drug Disc. Today: Technologies
Information 2006 | 3(3) | 307-313