2025

5
2025 6月
ERRα-Predictor: A Framework of Ensemble Models for Prediction of ERRα Binders, Antagonists, and Agonists Using Artificial Intelligence
作者: Le Xiong, Jiahao Xu, Hongbo Yu, Weihua Li, Xinmin Li, Wenxiang Song, Jingwei Zhang, Yun Tang*, Guixia Liu*
期刊: Journal of Chemical Information and Modeling
信息: 2025 | 65(13) | 6809–6822
2025 6月
In Silico Prediction of pKa Values Using Explainable Deep Learning Methods
作者: Chen Yang, Changda Gong, Zhixing Zhang, Jiaojiao Fang, Weihua Li, Guixia Liu, Yun Tang
期刊: Journal of Pharmaceutical Analysis
信息: 2025 | 15(6) | 101174
2025 4月
TCnet: a novel strategy to predict target combination of Alzheimer’s disease via network-based methods
作者: Yue CY, Chen BY, Pan F, Wang Z, Yu HB, Liu GX, Li WH, Wang R*, Tang Y*
期刊: Journal of Chemical Information and Modeling
信息: 2025
2025 3月
Cocry-pred: a dynamic resource propagation method for cocrystal prediction
作者: Song WX#, Peng R#, Yu HB, Zhan ML, Liu GX, Li WH, Ren GB, Zhu B*, Tang Y*
期刊: Journal of Chemical Information and Modeling
信息: 2025 | 65(6) | 2868-2881
2025 3月
Fluor-Predictor: An Interpretable Tool for Multiproperty Prediction and Retrieval of Fluorescent Dyes
作者: Wenxiang Song, Le Xiong, Xinmin Li, Yuyang Zhang, Binya Wang, Guixia Liu, Weihua Li, Youjun Yang*, Yun Tang*
期刊: Journal of Chemical Information and Modeling
信息: 2025 | 65(6) | 2868–2881

2024

4
2024 11月
ToxGIN: an In silico prediction model for peptide toxicity via graph isomorphism networks integrating peptide sequence and structure information
作者: Qiule Yu, Zhixing Zhang, Guixia Liu, Weihua Li, Yun Tang*
期刊: Briefings in Bioinformatics
信息: 2024 | 25(6) | bbae583
2024 10月
In Silico Prediction of ERRα Agonists Based on Combined Features and Stacking Ensemble Method
作者: Jiahao Xu, Zejun Huang, Hao Duan, Weihua Li, Jingyan Zhuang, Le Xiong, Yun Tang, Guixia Liu
期刊: ChemMedChem
信息: 2024 | 19(20) | e202400298
2024 6月
人工智能在抗癌肽研发中的应用与挑战
作者: Zhixing Zhang, Hua Deng, Yun Tang
期刊: 中国药科大学学报
信息: 2024 | Vol.55(3) | 347 − 356
2024 3月
MedChatZH: A tuning LLM for traditional Chinese medicine consultations
作者: Yang Tan, Zhixing Zhang, Mingchen Li, Fei Pan, Hao Duan, Zijie Huang, Hua Deng, Zhuohang Yu, Chen Yang, Guoyang Shen, Peng Qi, Chengyuan Yue, Yuxian Liu, Liang Hong, Huiqun Yu, Guisheng Fan, Yun Tang
期刊: Computers in Biology and Medicine
信息: 2024 | Vol.172 | 108290

2022

16
2022 12月
Development of In Silico Models for Predicting Potential Time-Dependent Inhibitors of Cytochrome P450 3A4
作者: Minjie Xu, Zhou Lu, Zengrui Wu, Minyan Gui, Guixia Liu, Yun Tang*, Weihua Li*
期刊: Molecular Pharmaceutics
信息: 2022 | 20(1) | 194–205
2022 11月
In silico prediction of chemical aquatic toxicity by multiple machine learning and deep learning approaches
作者: Minjie Xu, Hongbin Yang, Guixia Liu, Yun Tang, Weihua Li*
期刊: Journal of Applied Toxicology
信息: 2022 | 42(11) | 1766-1776
2022 10月
In silico prediction of potential drug-induced nephrotoxicity with machine learning methods
作者: Yuning Gong, Dan Teng, Yimeng Wang, Yaxin Gu, Zengrui Wu, Weihua Li, Yun Tang*, Guixia Liu*
期刊: Journal of Applied Toxicology
信息: 2022 | 42(10) | 1639-1650
2022 9月
In Silico Prediction of Human and Rat Liver Microsomal Stability via Machine Learning Methods
作者: Longqiang Li, Zhou Lu, Guixia Liu, Yun Tang, Weihua Li*
期刊: Chemical Research in Toxicology
信息: 2022 | 35(9) | 1614–1624
2022 9月
Profiling prediction of nuclear receptor modulators with multi-task deep learning methods: toward the virtual screening
作者: Jiye Wang, Chaofeng Lou, Guixia Liu, Weihua Li, Zengrui Wu, Yun Tang*
期刊: Briefings in Bioinformatics
信息: 2022 | 23(5) | bbac351
2022 9月
Drug Repurposing for Newly Emerged Diseases via Network-based Inference on a Gene-disease-drug Network
作者: Li Qin, Jiye Wang, Zengrui Wu, Weihua Li, Guixia Liu, Yun Tang*
期刊: Molecular Informatics
信息: 2022 | 41(9) | e2200001
2022 8月
Prediction of anti-inflammatory peptides by a sequence-based stacking ensemble model named AIPStack
作者: Hua Deng, Chaofeng Lou, Zengrui Wu, Weihua Li, Guixia Liu, Yun Tang*
期刊: iScience
信息: 2022 | 25(9) | 104967
2022 7月
Mechanistic Studies on the Stereoselectivity of FFAR1 Modulators
作者: Dan Teng, Yang Zhou, Yun Tang, Guixia Liu*, Yaoquan Tu*
期刊: Journal of Chemical Information and Modeling
信息: 2022 | 61(15) | 3664–3675
2022 7月
In silico prediction of UGT-mediated metabolism in drug-like molecules via graph neural network
作者: Mengting Huang, Chaofeng Lou, Zengrui Wu, Weihua Li, Philip W. Lee, Yun Tang*, Guixia Liu*
期刊: Journal of Cheminformatics
信息: 2022
2022 6月
Investigation of the mechanism of Shen Qi Wan prescription in the treatment of T2DM via network pharmacology and molecular docking
作者: Piaopiao Zhao, Xiaoxiao Zhang, Yuning Gong, Weihua Li, Zengrui Wu, Yun Tang*, Guixia Liu*
期刊: in Silico Pharmacology
信息: 2022 | 10(9)
2022 5月
IDL-PPBopt: A Strategy for Prediction and Optimization of Human Plasma Protein Binding of Compounds via an Interpretable Deep Learning Method
作者: Chaofeng Lou, Hongbin Yang, Jiye Wang, Mengting Huang, Weihua Li, Guixia Liu, Philip W. Lee, Yun Tang*
期刊: Journal of Chemical Information and Modeling
信息: 2022 | 62(11) | 2788–2799
2022 3月
A multitask GNN-based interpretable model for discovery of selective JAK inhibitors
作者: Yimeng Wang, Yaxin Gu, Chaofeng Lou, Yuning Gong, Zengrui Wu, Weihua Li, Yun Tang*, Guixia Liu*
期刊: Journal of Cheminformatics
信息: 2022 | 14(1) | 16
2022 3月
ADENet: a novel network-based inference method for prediction of drug adverse events
作者: Zhuohang Yu, Zengrui Wu*, Weihua Li, Guixia Liu, Yun Tang*
期刊: Briefings in Bioinformatics
信息: 2022 | 23(2) | bbab580
2022 2月
In Silico Prediction of Potential Drug Combinations for Type 2 Diabetes Mellitus by an Integrated Network and Transcriptome Analysis
作者: Dan Teng, Yuning Gong, Zengrui Wu, Weihua Li, Yun Tang*, Guixia Liu*
期刊: Chemmedchem
信息: 2022 | 17(3) | e202100620
2022 1月
wSDTNBI: a novel network-based inference method for virtual screening
作者: Zengrui Wu#, Hui Ma#, Zehui Liu#, Lulu Zheng, Zhuohang Yu, Shuying Cao, Wenqing Fang, Lili Wu, Weihua Li, Guixia Liu, Jin Huang, Yun Tang*
期刊: Chemical Science
信息: 2022 | 13(4) | 1060-1079
2022 1月
Discovery of New Estrogen-Related Receptor α Agonists via a Combination Strategy Based on Shape Screening and Ensemble Docking
作者: Dongping Li, Kexin Jiang, Dan Teng, Zengrui Wu, Weihua Li, Yun Tang*, Rui Wang*, Guixia Liu*
期刊: Journal of Chemical Information and Modeling
信息: 2022 | 62(3) | 486–497

2021

9
2021
Insights into the Molecular Mechanisms of Liuwei Dihuang Decoction via Network Pharmacology
作者: Jianhui Chen, Dan Teng, Zengrui Wu, Weihua Li, Yuqian Feng, Yun Tang*, Guixia Liu*
期刊: Chem. Res. Toxicol.
信息: 2021 | 34(1) | 91-102
2021
In silico prediction of chemical acute contact toxicity on honey bees via machine learning methods
作者: Xuan Xu, Piaopiao Zhao, Zhiyuan Wang, Xiaoxiao Zhang, Zengrui Wu, Weihua Li, Yun Tang*, Guixia Liu*
期刊: Toxicol. In Vitro
信息: 2021 | Vol.72 | 105089
2021
In silico prediction of mitochondrial toxicity of chemicals using machine learning methods
作者: Piaopiao Zhao, Yayuan Peng, Xuan Xu, Zhiyuan Wang, Zengrui Wu, Weihua Li, Yun Tang*, Guixia Liu*
期刊: J. Appl. Toxicol.
信息: 2021 | Vol.DOI | 10
2021
In silico prediction of chemical respiratory toxicity via machine learning
作者: Zhiyuan Wang, Piaopiao Zhao, Xiaoxiao Zhang, Xuan Xu, Weihua Li, Guixia Liu, Yun Tang*
期刊: Comput. Toxicol.
信息: 2021 | Vol.18 | 100155
2021
Assessment of CYP2C9 Structural Models for Site of Metabolism Prediction
作者: Xiaoxiao Zhang, Minjie Xu, Zengrui Wu, Guixia Liu, Yun Tang, Weihua Li*
期刊: ChemMedChem
信息: 2021 | Vol.DOI | 10
2021
Twin drug design, synthesis and evaluation of diosgenin derivatives as multitargeted agents for the treatment of vascular dementia
作者: Guixiang Yang, Jiamin Sun, Lulu Zheng, Li Zhang, Jie Li, Haixian Gan, Yan Huang, Jin Huang, Xingxing Diao, Yun Tang*, Rui Wang*, Lei Ma*
期刊: Bioorg. Med. Chem.
信息: 2021 | Vol.37 | 116109
2021
Homotropic Cooperativity of Midazolam Metabolism by Cytochrome P450 3A4: Insight from Computational Studies
作者: Junhao Li, Yue Chen, Yun Tang, Weihua Li*, Yaoquan Tu*
期刊: J. Chem. Inf. Model.
信息: 2021 | 61(5) | 2418-2426
2021
Pathway-Based Drug Repurposing with DPNetinfer: A Method to Predict Drug–Pathway Associations via Network-Based Approaches
作者: Jiye Wang, Zengrui Wu, Yayuan Peng, Weihua Li, Guixia Liu, Yun Tang*
期刊: J. Chem. Inf. Model.
信息: 2021 | 61(5) | 2475-2485
2021
Discovery of Natural Products Targeting NQO1 via an Approach Combining Network-Based Inference and Identification of Privileged Substructures
作者: Zengrui Wu, Qiaohui Wang, Hongbin Yang, Jiye Wang, Weihua Li, Guixia Liu, Yi Yang, Yuzheng Zhao*, Yun Tang*
期刊: J. Chem. Inf. Model.
信息: 2021 | 61(5) | 2486-2498

2020

14
2020
In Silico Prediction of Human Renal Clearance of Compounds Using Quantitative Structure-Pharmacokinetic Relationship Models
作者: Jianhui Chen, Hongbin Yang, Lan Zhu, Zengrui Wu, Weihua Li, Yun Tang*, Guixia Liu*
期刊: Chem. Res. Toxicol.
信息: 2020 | 33(2) | 640-650
2020
Mechanistic Insights into the Regio- and Stereoselectivities of Testosterone and Dihydrotestosterone Hydroxylation Catalyzed by CYP3A4 and CYP19A1
作者: Junhao Li, Yun Tang, Weihua Li*, Yaoquan Tu*
期刊: Chem. - Eur. J.
信息: 2020 | 26(28) | 6214-6223
2020
Computational Approaches to Identify Structural Alerts and Their Applications in Environmental Toxicology and Drug Discovery
作者: Hongbin Yang, Chaofeng Lou, Weihua Li, Guixia Liu, Yun Tang*
期刊: Chem. Res. Toxicol.
信息: 2020 | 33(6) | 1312-1322
2020
Computational Insight into the Allosteric Activation Mechanism of Farnesoid X Receptor
作者: Yue Chen, Junhao Li, Zengrui Wu, Guixia Liu, Honglin Li, Yun Tang*, Weihua Li*
期刊: J. Chem. Inf. Model.
信息: 2020 | 60(3) | 1540-1550
2020
In Silico Prediction of Metabolic Epoxidation for Drug-like Molecules via Machine Learning Methods
作者: Jiajing Hu, Yingchun Cai, Weihua Li, Guixia Liu, Yun Tang*
期刊: Mol. Inf.
信息: 2020 | 39(8) | 1900178
2020
In silico prediction of binding capacity and interaction forces of organic compounds with α- and β-cyclodextrins
作者: Peiwen Di, Jianhui Chen, Liping Liu, Weihua Li, Yun Tang*, Guixia Liu*
期刊: J. Mol. Liq.
信息: 2020 | Vol.302 | 112585
2020
Drug repositioning by prediction of drug's anatomical therapeutic chemical code via network-based inference approaches
作者: Yayuan Peng, Manjiong Wang, Yixiang Xu, Zengrui Wu, Jiye Wang, Chao Zhang, Guixia Liu, Weihua Li, Jian Li*, Yun Tang*
期刊: Briefings Bioinf.
信息: 2020 | 22(2) | 2058–2072
2020
Computational Insights into Molecular Activation and Positive Cooperative Mechanisms of FFAR1 Modulators
作者: Dan Teng, Jianhui Chen, Dongping Li, Zengrui Wu, Weihua Li, Yun Tang*, Guixia Liu*
期刊: J. Chem. Inf. Model.
信息: 2020 | 60(6) | 3214-3230
2020
In silico prediction of chemical neurotoxicity using machine learning
作者: Changsheng Jiang, Piaopiao Zhao, Weihua Li, Yun Tang*, Guixia Liu*
期刊: Toxicol. Res.
信息: 2020 | 9(3) | 164–172
2020
NetInfer: A Web Server for Prediction of Targets and Therapeutic and Adverse Effects via Network-Based Inference Methods
作者: Zengrui Wu, Yayuan Peng, Zhuohang Yu, Weihua Li, Guixia Liu, Yun Tang*
期刊: J. Chem. Inf. Model.
信息: 2020 | 60(8) | 3687-3691
2020
Dissecting the Structural Plasticity and Dynamics of Cytochrome P450 2B4 by Molecular Dynamics Simulations
作者: Junhao Li, Yang Zhou, Yun Tang, Weihua Li*, Yaoquan Tu*
期刊: J. Chem. Inf. Model.
信息: 2020 | 60(10) | 5026-5035
2020
Strategy for Efficient Discovery of Cocrystals via a Network-Based Recommendation Model
作者: Lulu Zheng, Bin Zhu, Zengrui Wu, Xiaoxue Fang, Minghuang Hong, Guixia Liu, Weihua Li, Guobin Ren*, Yun Tang*
期刊: Cryst. Growth Des.
信息: 2020 | 20(10) | 6820-6830
2020
Insights into the mechanism of Arnebia euchroma on leukemia via network pharmacology approach
作者: Biting Wang, Zengrui Wu*, Jiye Wang, Weihua Li, Guixia Liu, Bo Zhang, Yun Tang*
期刊: BMC Complementary Med. Ther.
信息: 2020 | 20(1) | 322
2020
MetaADEDB 2
作者: Zhuohang Yu, Zengrui Wu*, Weihua Li, Guixia Liu, Yun Tang*
期刊: 0: a comprehensive database on adverse drug events. Bioinformatics
信息: 2020 | Vol.DOI | 10

2019

13
2019
Computational Prediction of Site of Metabolism for UGT-Catalyzed Reactions
作者: Yingchun Cai, Hongbin Yang, Weihua Li, Guixia Liu, Philip W Lee, Yun Tang*
期刊: J. Chem. Inf. Model.
信息: 2019 | 59(3) | 1085-1095
2019
Computational insights into the different catalytic activities of CYP3A4 and CYP3A5 toward schisantherin E
作者: Yuhan Xue, Junhao Li, Zengrui Wu, Guixia Liu, Yun Tang, Weihua Li*
期刊: Chem. Biol. Drug Des.
信息: 2019 | 93(5) | 854–864
2019
In silico prediction of chemical reproductive toxicity using machine learning
作者: Changsheng Jiang, Hongbin Yang, Peiwen Di, Weihua Li, Yun Tang*, Guixia Liu*
期刊: J. Appl. Toxicol.
信息: 2019 | 39(6) | 844-854
2019
Computational insights into the interaction mechanisms of estrogen-related receptor alpha with endogenous ligand cholesterol
作者: Dongping Li, Yingchun Cai, Dan Teng, Weihua Li, Yun Tang*, Guixia Liu*
期刊: Chem. Biol. Drug Des.
信息: 2019 | 94(1) | 1316-1329
2019
In Silico Prediction of Endocrine Disrupting Chemicals Using Single-Label and Multilabel Models
作者: Lixia Sun, Hongbin Yang, Yingchun Cai, Weihua Li, Guixia Liu, Yun Tang*
期刊: J. Chem. Inf. Model.
信息: 2019 | 59(3) | 973-982
2019
Insights into the antineoplastic mechanism of Chelidonium majus via systems pharmacology approach
作者: Xinzhe Xiao, Zehui Chen, Zengrui Wu, Tianduanyi Wang, Weihua Li, Guixia Liu, Bo Zhang*, Yun Tang*
期刊: Quant. Biol.
信息: 2019 | 7(1) | 42-53
2019
Prediction of the skin sensitising potential and potency of compounds via mechanism-based binary and ternary classification models
作者: Peiwen Di, Yongmin Yin, Changsheng Jiang, Yingchun Cai, Weihua Li, Yun Tang*, Guixia Liu*
期刊: Toxicol. In Vitro
信息: 2019 | Vol.59 | 204-214
2019
Insights into mechanisms and severity of drug-induced liver injury via computational systems toxicology approach
作者: Yayuan Peng, Zengrui Wu*, Hongbin Yang, Yingchun Cai, Guixia Liu, Weihua Li, Yun Tang*
期刊: Toxicol. Lett.
信息: 2019 | Vol.312 | 22-33
2019
A novel derivative of artemisinin inhibits cell proliferation and metastasis via down-regulation of cathepsin K in breast cancer
作者: Xiangyu Gu, Yayuan Peng, Yuyu Zhao, Xin Liang*, Yun Tang*, Jianwen Liu*
期刊: Eur. J. Pharmacol.
信息: 2019 | Vol.858 | 172382
2019
Design, synthesis and biological evaluation of chalcones as reversers of P-glycoprotein-mediated multidrug resistance
作者: Huanhuan Yin, Jingjing Dong, Yingchun Cai, Ximeng Shi, Hao Wang, Guixia Liu, Yun Tang*, Jianwen Liu*, Lei Ma*
期刊: Eur. J. Med. Chem.
信息: 2019 | Vol.180 | 350-366
2019
Prediction of the allergic mechanism of haptens via a reaction-substructure-compound-target-pathway network system
作者: Peiwen Di, Zengrui Wu, Hongbin Yang, Weihua Li, Yun Tang*, Guixia Liu*
期刊: Toxicol. Lett.
信息: 2019 | Vol.317 | 68-81
2019
Insights into the interaction mechanisms of estrogen-related receptor alpha (ERRα) with ligands via molecular dynamics simulations
作者: Dongping Li, Yingchun Cai, Dan Teng, Zengrui Wu, Weihua Li, Yun Tang*, Guixia Liu*
期刊: J. Biomol. Struct. Dyn.
信息: 2019 | 38(13) | 3867-3878
2019
Design, synthesis and evaluation of diosgenin carbamate derivatives as multitarget anti-Alzheimer's disease agents
作者: Guixiang Yang, Yan Huang, Lulu Zheng, Li Zhang, Lin Su, Yuhang Wu, Jie Li, Licheng Zhou, Jin Huang, Yun Tang*, Rui Wang*, Lei Ma*
期刊: Eur. J. Med. Chem.
信息: 2019 | Vol.187 | 111913

2018

14
2018
In Silico Prediction of Chemical Toxicity for Drug Design Using Machine Learning Methods and Structural Alerts
作者: Hongbin Yang, Lixia Sun, Weihua Li, Guixia Liu, Yun Tang*
期刊: Front. Chem.
信息: 2018 | Vol.6 | 30
2018
Corrigendum: In Silico Prediction of Chemical Toxicity for Drug Design Using Machine Learning Methods and Structural Alerts
作者: Hongbin Yang, Lixia Sun, Weihua Li, Guixia Liu, Yun Tang*
期刊: Front. Chem.
信息: 2018 | Vol.6 | 129
2018
Lee, Yun Tang*
作者: Yingchun Cai, Hongbin Yang, Weihua Li, Guixia Liu, Philip W
期刊: Multiclassification Prediction of Enzymatic Reactions for Oxidoreductases and Hydrolases Using Reaction Fingerprints and Machine Learning Methods. J. Chem. Inf. Model.
信息: 2018 | 58(6) | 1169-1181
2018
A Computational Systems Pharmacology Approach to Investigate Molecular Mechanisms of Herbal Formula Tian-Ma-Gou-Teng-Yin for Treatment of Alzheimer's Disease
作者: Tianduanyi Wang, Zengrui Wu, Lixia Sun, Weihua Li, Guixia Liu, Yun Tang*
期刊: Front. Chem.
信息: 2018 | Vol.9 | 668
2018
Identification of Nontoxic Substructures: A New Strategy to Avoid Potential Toxicity Risk
作者: Hongbin Yang, Lixia Sun, Weihua Li, Guixia Liu, Yun Tang*
期刊: Toxicol. Sci.
信息: 2018 | 165(2) | 396–407
2018
In silico estimation of chemical aquatic toxicity on crustaceans using chemical category methods
作者: Qianqian Cao, Lin Liu, Hongbin Yang, Yingchun Cai, Weihua Li, Guixia Liu, Philip W Lee, Yun Tang*
期刊: Environ. Sci.: Processes Impacts
信息: 2018 | 20(9) | 1234-1243
2018
In Silico Prediction of Blood–Brain Barrier Permeability of Compounds by Machine Learning and Resampling Methods
作者: Zhuang Wang, Hongbin Yang, Zengrui Wu, Tianduanyi Wang, Weihua Li, Yun Tang*, Guixia Liu*
期刊: ChemMedChem.
信息: 2018 | 13(20) | 2189–2201
2018
admetSAR 2
作者: Hongbin Yang, Chaofeng Lou, Lixia Sun, Jie Li, Yingchun Cai, Zhuang Wang, Weihua Li, Guixia Liu, Yun Tang*
期刊: 0: web-service for prediction and optimization of chemical ADMET properties. Bioinformatics.
信息: 2018 | 35(6) | 1067-1069
2018
Computational Insight Into Vitamin K1 ω-Hydroxylation by Cytochrome P450 4F2
作者: Junhao Li, Hongxiao Zhang, Guixia Liu, Yun Tang, Yaoquan Tu*, Weihua Li*
期刊: Front. Pharmacol.
信息: 2018 | Vol.9 | 1065
2018
ADMETopt: A Web Server for ADMET Optimization in Drug Design via Scaffold Hopping
作者: Hongbin Yang, Lixia Sun, Zhuang Wang, Weihua Li, Guixia Liu, Yun Tang*
期刊: J. Chem. Inf. Model.
信息: 2018 | 58(10) | 2051-2056
2018
Network-Based Methods for Prediction of Drug-Target Interactions
作者: Zengrui Wu, Weihua Li, Guixia Liu, Yun Tang*
期刊: Front. Pharmacol.
信息: 2018 | Vol.9 | 1134
2018
Prediction of Farnesoid X Receptor Disruptors with Machine Learning Methods
作者: Yue Chen, Hongbin Yang, Zengrui Wu, Guixia Liu, Yun Tang, Weihua Li*
期刊: Chem. Res. Toxicol.
信息: 2018 | 31(11) | 1128-1137
2018
ADMET-score – a comprehensive scoring function for evaluation of chemical drug-likeness
作者: Longfei Guan, Hongbin Yang, Yingchun Cai, Lixia Sun, Peiwen Di, Weihua Li, Guixia Liu, Yun Tang*
期刊: MedChemComm.
信息: 2018 | 10(1) | 148-157
2018
Modified rivaroxaban microparticles for solid state properties improvement based on drug-protein/polymer supramolecular interactions
作者: Ning Chen, Peiwen Di, Shangqi Ning, Wenjun Jiang, Qiufang Jing, Guobin Ren, Yan Liu, Yun Tang, Zhongyu Xu, Guixia Liu*, Fuzheng Ren*
期刊: Powder Technol.
信息: 2018 | Vol.344 | 819–829

2017

14
2017
Computational Investigation of Ligand Binding to the Peripheral Site in CYP3A4: Conformational Dynamics and Inhibitor Discovery
作者: Hanwen Du, Junhao Li, Yingchun Cai, Hongxiao Zhang, Guixia Liu, Yun Tang*, Weihua Li*
期刊: J. Chem. Inf. Model.
信息: 2017 | 57(3) | 616-626
2017
Insights into the molecular mechanisms of Polygonum multiflorum Thunb-induced liver injury: a computational systems toxicology approach
作者: Yinyin Wang, Jie Li, Zengrui Wu, Bo Zhang, Hongbin Yang, Qin Wang, Yingchun Cai, Guixia Liu, Weihua Li, Yun Tang*
期刊: Acta Pharmacol. Sin.
信息: 2017 | 38(5) | 719-732
2017
In Silico Prediction of Chemicals Binding to Aromatase with Machine Learning Methods
作者: Hanwen Du, Yingchun Cai, Hongbin Yang, Hongxiao Zhang, Yuhan Xue, Guixia Liu, Yun Tang, Weihua Li*
期刊: Chem. Res. Toxicol.
信息: 2017 | 30(5) | 1209-1218
2017
Improving the physicochemical properties of bicalutamide by complex formation with bovine serum albumin
作者: Congbin Yang, Peiwen Di, Jinping Fu, Hui Xiong, Qiufang Jing, Guobin Ren, Yun Tang, Wenyun Zheng, Guixia Liu*, Fuzheng Ren*
期刊: Eur. J. Pharm. Sci.
信息: 2017 | Vol.106 | 381-392
2017
Evaluation of Different Methods for Identification of Structural Alerts Using Chemical Ames Mutagenicity Data Set as a Benchmark
作者: Hongbin Yang, Jie Li, Zengrui Wu, Weihua Li, Guixia Liu, Yun Tang*
期刊: Chem. Res. Toxicol.
信息: 2017 | 30(6) | 1355-1364
2017
In silico prediction of chemical subcellular localization via multi-classification methods
作者: Hongbin Yang, Xiao Li, Yingchun Cai, Qin Wang, Weihua Li, Guixia Liu, Yun Tang*
期刊: MedChemComm.
信息: 2017 | 8(6) | 1225-1234
2017
In silico prediction of pesticide aquatic toxicity with chemical category approaches
作者: Fuxing Li, Defang Fan, Hao Wang, Hongbin Yang, Weihua Li, Yun Tang*, Guixia Liu*
期刊: Toxicol. Res.
信息: 2017 | 6(6) | 831–842
2017
Quantitative and Systems Pharmacology
作者: Jiansong Fang, Zengrui Wu, Chuipu Cai, Qi Wang, Yun Tang*, Feixiong Cheng*
期刊: 1. In Silico Prediction of Drug–Target Interactions of Natural Products Enables New Targeted Cancer Therapy. J. Chem. Inf. Model.
信息: 2017 | 57(11) | 2657-2671
2017
In Silico Prediction of Compounds Binding to Human Plasma Proteins by QSAR Models
作者: Lixia Sun, Hongbin Yang, Jie Li, Tianduanyi Wang, Weihua Li, Guixia Liu, Yun Tang*
期刊: ChemMedChem.
信息: 2017 | 13(6) | 572–581
2017
Computational insights into the subtype selectivity and “message-address-efficacy” mechanisms of opioid receptors through JDTic binding and unbinding
作者: Jianxin Cheng, Tao Cheng, Weihua Li, Guixia Liu, Weiliang Zhu, Yun Tang*
期刊: Acta Pharmacol. Sin.
信息: 2017 | 39(3) | 482-491
2017
Quantitative and systems pharmacology 2
作者: Zengrui Wu, Weiqiang Lu, Weiwei Yu, Tianduanyi Wang, Weihua Li, Guixia Liu, Hankun Zhang, Xiufeng Pang, Jin Huang, Mingyao Liu*, Feixiong Cheng*, Yun Tang*
期刊: In silico polypharmacology of G protein-coupled receptor ligands via network-based approaches. Pharmacol. Res.
信息: 2017 | Vol.129 | 400-413
2017
Computational insights into the G-protein-biased activation and inactivation mechanisms of the μ opioid receptor
作者: Jianxin Cheng, Tao Cheng, Weihua Li, Guixia Liu, Weiliang Zhu, Yun Tang*
期刊: Acta Pharmacol. Sin.
信息: 2017 | 39(1) | 154-164
2017
Network pharmacological mechanisms of Vernonia anthelmintica (L
作者: Jiye Wang, Hong Chen, Yinyin Wang, Xiaoqin Wang, Hanying Chen, Mei Zhang, Yun Tang*, Bo Zhang*
期刊: ) in the treatment of vitiligo: Isorhamnetin induction of melanogenesis via up-regulation of melanin-biosynthetic genes. BMC Syst. Biol.
信息: 2017 | 11(1) | 103
2017
In silico prediction of chemical genotoxicity using machine learning methods and structural alerts
作者: Defang Fan, Hongbin Yang, Fuxing Li, Lixia Sun, Peiwen Di, Weihua Li, Yun Tang*, Guixia Liu*
期刊: Toxicol. Res.
信息: 2017 | 7(2) | 211-220

2016

9
2016
Effects of protein flexibility and active site water molecules on the prediction of sites of metabolism for cytochrome P450 2C19 substrates
作者: Junhao Li, Jinya Cai, Haixia Su, Hanwen Du, Juan Zhang, Shihui Ding, Guixia Liu, Yun Tang*, Weihua Li*
期刊: Mol. BioSyst.
信息: 2016 | 12(3) | 868-878
2016
Lee, Yun Tang*
作者: Chen Zhang, Yuan Zhou, Shikai Gu, Zengrui Wu, Wenjie Wu, Changming Liu, Kaidong Wang, Guixia Liu, Weihua Li, Philip W
期刊: In silico prediction of hERG potassium channel blockage by chemical category approaches. Toxicol. Res.
信息: 2016 | 5(2) | 570-582
2016
Computational insight into conformational states of glucagon-like peptide-1 receptor (GLP-1R) and its binding mode with GLP-1
作者: Juan Zhang, Shikai Gu, Xianqiang Sun, Weihua Li, Yun Tang*, Guixia Liu*
期刊: RSC Adv.
信息: 2016 | 6(16) | 13490-13497
2016
Computational insights into different inhibition modes of the κ-opioid receptor with antagonists LY2456302 and JDTic
作者: Jianxin Cheng, Weihua Li, Guixia Liu, Weiliang Zhu, Yun Tang*
期刊: RSC Adv.
信息: 2016 | 6(17) | 13626-13635
2016
SDTNBI: an integrated network and chemoinformatics tool for systematic prediction of drug–target interactions and drug repositioning
作者: Zengrui Wu, Feixiong Cheng, Jie Li, Weihua Li, Guixia Liu, Yun Tang*
期刊: Brief Bioinform.
信息: 2016 | Vol.DOI | 10
2016
Interactions of omeprazole-based analogues with cytochrome P450 2C19: a computational study
作者: Junhao Li, Hanwen Du, Zengrui Wu, Haixia Su, Guixia Liu, Yun Tang*, Weihua Li*
期刊: Mol. BioSyst.
信息: 2016 | 12(6) | 1913-1921
2016
Network-based identification of microRNAs as potential pharmacogenomic biomarkers for anticancer drugs
作者: Jie Li, Kecheng Lei, Zengrui Wu, Weihua Li, Guixia Liu, Jianwen Liu, Feixiong Cheng, Yun Tang*
期刊: Oncotarget
信息: 2016 | 7(29) | 45584-45596
2016
In silico prediction of chemical mechanism of action via an improved network-based inference method
作者: Zengrui Wu, Weiqiang Lu, Dang Wu, Anqi Luo, Hanping Bian, Jie Li, Weihua Li, Guixia Liu, Jin Huang*, Feixiong Cheng, Yun Tang*
期刊: Br. J. Pharmacol.
信息: 2016 | 173(23) | 3372-3385
2016
Computational investigation of the interaction mechanism between the estrogen related receptor α and its agonists
作者: Fuxing Li, Xianqiang Sun, Yingchun Cai, Defang Fan, Weihua Li, Yun Tang*, Guixia Liu*
期刊: RSC Adv.
信息: 2016 | 6(96) | 94119-94127

2015

10
2015
Lee*, Yun Tang*
作者: Chen Zhang, Feixiong Cheng, Lu Sun, Shulin Zhuang, Weihua Li, Guixia Liu, Philip W
期刊: In silico prediction of chemical toxicity on avian species using chemical category approaches. Chemosphere
信息: 2015 | Vol.122 | 280-287
2015
Discovery of New Non-Steroidal Farnesoid X Receptor Modulators Through 3D Shape Similarity Search and Structure-Based Virtual Screening
作者: Lei Wang, Pei Si, Yayun Sheng, Yingjie Chen, Ping Wan, Xu Shen, Yun Tang, Lili Chen*, Weihua Li*
期刊: Chem. Biol. Drug Des.
信息: 2015 | Vol.85 | 481-487
2015
Lee, Yun Tang*
作者: Lu Sun, Chen Zhang, Yingjie Chen, Xiao Li, Shulin Zhuang, Weihua Li, Guixia Liu, Philip W
期刊: In silico prediction of chemical aquatic toxicity with chemical category approaches and substructural alerts. Toxicol. Res.
信息: 2015 | Vol.4 | 452-463
2015
FXR antagonism of NSAIDs contributes to drug-induced liver injury identified by systems pharmacology approach
作者: Weiqiang Lu, Feixiong Cheng, Jing Jiang, Chen Zhang, Xiaokang Deng, Zhongyu Xu, Shien Zou*, Xu Shen, Yun Tang*, Jin Huang*
期刊: Scientific Reports
信息: 2015 | Vol.5 | 8114
2015
Residues remote from the binding pocket control the antagonist selectivity towards the corticotropin-releasing factor receptor-1
作者: Xianqiang Sun, Jianxin Cheng, Xu Wang, Yun Tang*, Hans Agren, Yaoquan Tu*
期刊: Scientific Reports
信息: 2015 | Vol.5 | 8066
2015
In Silico Estimation of Chemical Carcinogenicity with Binary and Ternary Classification Methods
作者: Xiao Li, Zheng Du, Jie Wang, Zengrui Wu, Weihua Li, Guixia Liu, Xu Shen, Yun Tang*
期刊: Mol. Inform.
信息: 2015 | Vol.34 | 228-235
2015
Quantitative Regression Models for the Prediction of Chemical Properties by an Efficient Workflow
作者: Yongmin Yin, Congying Xu, Shikai Gu, Weihua Li, Guixia Liu*, Yun Tang*
期刊: Mol. Inform.
信息: 2015 | 34(10) | 679-688
2015
Association between cigarette smoking and Parkinson's disease: A meta-analysis
作者: Xiao Li, Weihua Li, Guixia Liu, Xu Shen, Yun Tang*
期刊: Arch. Gerontol. Geriat.
信息: 2015 | 61(3) | 510-516
2015
Mendrick, Yun Tang*, Feixiong Cheng*
作者: Chen Zhang, Huixiao Hong, Donna L
期刊: Biomarker-based drug safety assessment in the age of systems pharmacology: from foundational to regulatory science. Biomark. Med.
信息: 2015 | 9(11) | 1241-1252
2015
Computational insights into inhibitory mechanism of azole compounds against human aromatase
作者: Jinya Cai, Junhao Li, Juan Zhang, Shihui Ding, Guixia Liu, Weihua Li*, Yun Tang*
期刊: RSC Adv.
信息: 2015 | 5(110) | 90871-90880

2014

6
2014
Computational prediction of microRNA networks incorporating environmental toxicity and disease etiology
作者: Jie Li, Zengrui Wu, Feixiong Cheng, Weihua Li, Guixia Liu, Yun Tang*
期刊: Scientific Reports
信息: 2014 | Vol.4 | 5576
2014
Selective ligands of estrogen receptor β discovered using pharmacophore mapping and structure-based virtual screening
作者: Lei Chen, Dang Wu, Hanping Bian, Guanglin Kuang, Jing Jiang, Weihua Li, Guixia Liu, Shien Zou*, Jin Huang, Yun Tang*
期刊: Acta Pharmacol. Sin.
信息: 2014 | Vol.35 | 1333-1341
2014
Structure-based ensemble-QSAR model: a novel approach to the study of the EGFR tyrosine kinase and its inhibitors
作者: Xianqiang Sun, Lei Chen, Yaozong Li, Weihua Li, Guixia Liu, Yaoquan Tu*, Yun Tang*
期刊: Acta Pharmacol. Sin.
信息: 2014 | Vol.35 | 301-310
2014
In Silico Prediction of Chemical Acute Oral Toxicity Using Multi-Classification Methods
作者: Xiao Li, Lei Chen, Feixiong Cheng, Zengrui Wu, Hanping Bian, Congying Xu, Weihua Li, Guixia Liu, Xu Shen, Yun Tang*
期刊: J. Chem. Inf. Model.
信息: 2014 | 54(4) | 1061-1069
2014
Effects of protein flexibility on the site of metabolism prediction for CYP2A6 substrates
作者: Yayun Sheng, Yingjie Chen, Lei Wang, Guixia Liu, Weihua Li*, Yun Tang*
期刊: J. Mol. Graph. Model.
信息: 2014 | Vol.54 | 90-99
2014
Computational models to predict endocrine-disrupting chemical binding with androgen or oestrogen receptors
作者: Yingjie Chen, Feixiong Cheng, Lu Sun, Weihua Li, Guixia Liu, Yun Tang*
期刊: Ecotox. Environ. Safe.
信息: 2014 | Vol.110 | 280-287

2013

8
2013
In Silico ADMET Prediction: Recent Advances, Current Challenges and Future Trends
作者: Feixiong Cheng, Weihua Li, Guixia Liu, Yun Tang*
期刊: Curr Top Med Chem
信息: 2013 | 13(11) | 1273-1289
2013
Adverse Drug Events: Database Construction and In Silico Prediction
作者: Feixiong Cheng, Weihua Li, Xichuan Wang, Yadi Zhou, Zengrui Wu, Jie Shen and Yun Tang
期刊: J. Chem. Inf. Model.
信息: 2013 | 53(4) | 744-752
2013
Lee, Yun Tang*
作者: Feixiong Cheng, Weihua Li, Yadi Zhou, Jie Li, Jie Shen, Philip W
期刊: Prediction of Human Genes and Diseases Targeted by Xenobiotics Using Predictive Toxicogenomics-Derived Models (PTDMs). Mol. BioSyst
信息: 2013 | 9(6) | 1316-1325
2013
Prediction of Polypharmacological Profiles of Drugs by the Integration of Chemical, Side Effects and Therapeutic Space
作者: Feixiong Cheng, Weihua Li, Zengrui Wu, Xichuan Wang, Chen Zhang, Jie Li, Guixia Liu and Yun Tang
期刊: J. Chem. Inf. Model.
信息: 2013 | 53(4) | 753-762
2013
The role of benzoic acid in proline-catalyzed asymmetric michael addition: A density functional theory study
作者: Hongwei Shi, Xiangui Huang, Guixia Liu*, Kunqian Yu, Congying Xu, Weihua Li, Bubing Zeng*, Yun Tang*
期刊: Int. J. Quantum. Chem.
信息: 2013 | 113(9) | 1339-1348
2013
Catalytic Mechanism of Cytochrome P450 2D6 for 4-Hydroxylation of Aripiprazole: A QM/MM Study
作者: Rongwei Shi, Weihua Li, Guixia Liu, Yun Tang*
期刊: Chinese J. Chem.
信息: 2013 | 31(9) | 1219-1227
2013
Design, synthesis and biological evaluation of organophosphorous-homodimers as dual binding site acetylcholinesterase inhibitors
作者: Ruliang Xie, Qianfei Zhao, Tao Zhang, Jing Fang , Xiangdong Mei, Jun Ning*, Yun Tang*
期刊: Bioorg. Med. Chem.
信息: 2013 | 21(1) | 278-282
2013
Computational insights into the binding modes of Sr-Rex with cofactor NADH/NAD+ and operator DNA
作者: Yanyan Chu, Weihua Li, Jianfeng Wang, Guixia Liu, Yun Tang*
期刊: J. Mol. Model.
信息: 2013 | 19(8) | 3143-3151

2012

19
2012
Novel triazolyl bis-amino acid derivatives readily synthesized via click chemistry as potential corrosion inhibitors for mild steel in HCl
作者: Qiong Deng, Hong-Wei Shi, Bao-Qin Chen, Xiao-Peng He, Guixia Liu, Yun Tang, Yi-Tao Long, Guo-Rong Chen
期刊: Corros. Sci.
信息: 2012 | Vol.57 | 220-227
2012
In Silico Investigation of Interactions between Human Cannabinoid Receptor-1 and Its Antagonists
作者: Guanglin Kuang, Guoping Hu, Xianqiang Sun, Weihua Li, Guixia Liu, Yun Tang*
期刊: J. Mol. Model.
信息: 2012 | 18(8) | 3831-3845
2012
Lee* and Yun Tang*
作者: Feixiong Cheng, Yutaka Ikenaga, Yadi Zhou, Yue Yu, Weihua Li, Jie Shen, Zheng Du, Lei Chen, Congyin Xu, Guixia Liu, Philip W
期刊: In Silico Assessment of Chemical Biodegradability. J. Chem. Inf. Model.
信息: 2012 | 52(3) | 655-669
2012
Investigation of indazole unbinding pathways in CYP2E1 by molecular dynamics simulations
作者: Zhonghua Shen, Feixiong Cheng, You Xu, Jing Fu, Wen Xiao, Jie Shen, Guixia Liu, Weihua Li*, and Yun Tang*
期刊: PLoS One
信息: 2012 | 7(3) | e33500
2012
Synthesis and biological evaluation of quinazoline and quinoline bearing 2,2,6,6-tetramethylpiperidine-N-oxyl as potential epidermal growth factor receptor (EGFR) tyrosine kinase inhibitors and EPR bio-probe agents
作者: Siyuan Li, Chunying Guo, Xianqiang Sun, Yaozong Li, Hongli Zhao, Dongmei Zhan, Minbo Lan*, Yun Tang*
期刊: Euro. J. Med. Chem.
信息: 2012 | Vol.49 | 271-278
2012
Prediction of Drug-Target Interactions and Drug Repositioning via Network-Based Inference
作者: Feixiong Cheng, Chuang Liu, Jing Jiang, Weiqiang Lu, Weihua Li, Guixia Liu, Weixing Zhou, Jin Huang, and Yun Tang*
期刊: PLoS Comput Biol
信息: 2012 | 8(5) | e1002503
2012
Discovery of novel EGFR tyrosine kinase inhibitors by structure-based virtual screening
作者: Siyuan Li, Xianqiang Sun, Hongli Zhao, Yun Tang*, Minbo Lan*
期刊: Bioorg. Med. Chem. Lett.
信息: 2012 | 22(12) | 4004-4009
2012
Discovery and Structure-Activity Analysis of Selective Estrogen Receptor Modulators via Similarity-Based Virtual Screening
作者: Jie Shen, Jing Jiang, Guanglin Kuang, Chengfang Tan, Guixia Liu, Jin Huang*, and Yun Tang*
期刊: Euro. J. Med. Chem.
信息: 2012 | Vol.54 | 188-196
2012
Performance Evaluation of 2D Fingerprint and 3D Shape Similarity Methods in Virtual Screening
作者: Guoping Hu, Guanglin Kuang, Wen Xiao, Weihua Li, Guixia Liu, Yun Tang*
期刊: J. Chem. Inf. Model
信息: 2012 | 52(5) | 1103-1113
2012
Prediction of Chemical-Protein Interactions: Multitarget-QSAR versus Computational Chemogenomic Methods
作者: Feixiong Cheng, Yadi Zhou, Jie Li, Weihua Li, Guixia Liu and Yun Tang*
期刊: Mol. BioSyst.
信息: 2012 | Vol.8 | 2373-2384
2012
Identification of diverse dipeptidyl peptidase IV inhibitors via structure-based virtual screening
作者: Cui Li, Weiqiang Lu, Chunhua Lu, Wen Xiao,Xu Shen, Jin Huang, Guixia Liu*, Yun Tang*
期刊: J. Mol. Model.
信息: 2012 | Vol.18 | 4033-4042
2012
Concise CuI-Catalyzed Azide-Alkyne 1,3-Dipolar Cycloaddition Reaction Ligation Remarkably Enhances the Corrosion Inhibitive Potency of Natural Amino Acids for Mild Steel in HCl
作者: Qiong Deng, Xiaopeng He, Hongwei Shi, Baoqin Chen, Guixia Liu, Yun Tang, Yitao Long, Guorong Chen, and Kaixian Chen
期刊: Ind. Eng. Chem. Res.
信息: 2012 | Vol.51 | 7160-7169
2012
Synthesis, Structure–Activity Relationship, and Pharmacophore Modeling Studies of Pyrazole-3-Carbohydrazone Derivatives as Dipeptidyl Peptidase IV Inhibitors
作者: Deyan Wu, Fangfang Jin, Weiqiang Lu, Jin Zhu, Cui Li, Wei Wang, Yun Tang, Hualiang Jiang, Jin Huang, Guixia Liu, and Jian Li
期刊: Chem. Biol. Drug. Des.
信息: 2012 | Vol.79 | 897-906
2012
Prediction of Chemical-Protein Interactions Network with Weighted Network-based Inference Method
作者: Feixiong Cheng, Yadi Zhou, Weihua Li, Guixia Liu and Yun Tang*
期刊: PLoS One
信息: 2012 | 7(7) | e41064
2012
Lee, and Yun Tang*
作者: Congying Xu, Feixiong Cheng, Lei Chen, Zheng Du, Weihua Li, Guixia Liu, Philip W
期刊: In Silico Prediction of Chemical Ames Mutagenicity. J. Chem. Inf. Model.
信息: 2012 | 52(11) | 2840-2847
2012
Discovery of Inhibitors to Block Interactions of HIV-1 Integrase with Human LEDGF/p75 via Structure-Based Virtual Screening and Bioassays
作者: Guoping Hu, Xi Li, Xuan Zhang, Yaozong Li, Lei Ma, Liumeng Yang, Guixia Liu, Weihua Li, Jin Huang, Xu Shen, Lihong Hu, Yongtang Zheng and Yun Tang*
期刊: J. Med. Chem.
信息: 2012 | Vol.55 | 10108-10117
2012
Identification of old drugs as potential inhibitors of HIV-1 integrase-human LEDGF/p75 interaction via molecular docking
作者: Guoping Hu, Xi Li, Xianqiang Sun, Weiqiang Lu Guixia Liu, Jin Huang, Xu Shen and Yun Tang
期刊: J. Mol. Model
信息: 2012 | Vol.18 | 4995-5003
2012
Unbinding pathways of GW4064 from human farnesoid X receptor as revealed by molecular dynamics simulations
作者: Weihua Li, Jing Fu, Feixiong Cheng, Mingyue Zheng, Jian Zhang, Guixia Liu, and Yun Tang*
期刊: J. Chem. Inf. Model.
信息: 2012 | 52(11) | 3043-3052
2012
Inhibitors of HIV-1 Integrase-Human LEDGF/p75 Interaction Identified from Natural Products via Virtual Screening
作者: Guoping Hu, Xi Li, Yaozong Li, Xianqiang Sun, Guixia Liu, Weihua Li, Jin Huang*, Xu Shen, Yun Tang
期刊: Chin. J. Chem.
信息: 2012 | 30(12) | 2752-2758

2011

13
2011
Insights into binding modes of 5-HT2c receptor antagonists with ligand-based and receptor-based methods
作者: Chunhua Lu, Fangfang Jin, Cui Li, Weihua Li, Guixia Liu*, Yun Tang*
期刊: J Mol Model
信息: 2011 | 17(10) | 2513-2523
2011
Insights into subtype selectivity of opioid agonists by ligand-based and structure-based methods
作者: Jianxin Cheng, Guixia Liu*, Jing Zhang, Zhejun Xu and Yun Tang*
期刊: J Mol Model.
信息: 2011 | Vol.17 | 477-493
2011
Crucial role of the first CXXC motif of human QSOX 1b in protein thiol oxidation
作者: Zheng Wenyun, Chu Yanyan, Yin Qin, Xu Lei, Yang Charles, Zhang Wenyao, Tang Yun*, Yang Yi*
期刊: J. Biochemistry
信息: 2011 | 149(3) | 293-300
2011
Computational investigation of interactions between human H2 receptor and its agonists
作者: Sun Xianqiang, Li Yaozong, Li Weihua, Xu Zhejun, Tang Yun*
期刊: J. Mol. Graph. Modelling
信息: 2011 | 29(5) | 693-701
2011
Identification of small molecular inhibitors for Ero1p by structure-based virtual screening
作者: Chu Yanyan, Chen Xianjun, Yang Yi*, Tang Yun*
期刊: Bioorg. Med. Chem. Lett.
信息: 2011 | 21(4) | 1118-1121
2011
Lee, Tang Yun*
作者: Cheng Feixiong, Shen Jie, Yu Yue, Li Weihua*, Liu Guixia, Philip W
期刊: In silico prediction of Tetrahymena pyriformis toxicity for diverse industrial chemicals with substructure pattern recognition and machine learning methods. Chemosphere
信息: 2011 | 82(11) | 1636-1643
2011
Exploring coumarin egress channels in human cytochrome P450 2A6 by random acceleration and steered molecular dynamics simulations
作者: Weihua Li, Jie Shen, Guixia Liu, Tang Yun*, Tyuji Hoshino*
期刊: Proteins
信息: 2011 | 79(1) | 271-281
2011
Possible Ligand Release Pathway of Dipeptidyl Peptidase IV Investigated by Molecular Dynamics Simulations
作者: Cui Li, Jie Shen, Weihua Li, Chunhua Lu, Guixia Liu*, Yun Tang*
期刊: Proteins: Structure, Function and Bioinformatics.
信息: 2011 | 79(6) | 1800-1809
2011
Lee, and Yun Tang*
作者: Feixiong Cheng, Yue Yu, Jie Shen, Lei Yang, Weihua Li*, Guixia Liu, Philip W
期刊: Classification of Cytochrome P450 Inhibitors and non-Inhibitors using Combined Classifiers. J. Chem. Inf. Model.
信息: 2011 | 51(5) | 996-1011
2011
Computational insights into the different catalytic activities of CYP2A13 and CYP2A6 on NNK
作者: You Xu, Zhonghua Shen, Jie Shen, Guixia Liu, Weihua Li*, and Yun Tang*
期刊: J. Mol. Graph. Model.
信息: 2011 | Vol.30 | 1-9
2011
Computational Insights into Ligand Selectivity of Estrogen Receprors from Pharmacophore Modeling
作者: Jing Fang, Jie Shen, Feixiong Cheng, Zhejun Xu, Guixia Liu, and Yun Tang*
期刊: Mol. Inf.
信息: 2011 | Vol.30 | 539-549
2011
An Unusual (R)-Selective Epoxide Hydrolase with High Activity for Facile Preparation of Enantiopure Glycidyl Ethers
作者: Jing Zhao, Yan-Yan Chu, Ai-Tao Li, Xin Ju, Xu-Dong Kong, Jiang Pan, Yun Tang* and Jian-He Xu*
期刊: Adv. Synth. Catal.
信息: 2011 | Vol.353 | 1510-1518
2011
Click to a focused library of benzyl 6-triazolo(hydroxy)benzoic glucosides: Novel construction of PTP1B inhibitors on a sugar scaffold
作者: Cui Li, Xiao-Peng He, Yin-Jie Zhang, Zhen Li, Li-Xin Gao, Xiao-Xin Shi, Juan Xie, Jia Li, Guo-Rong Chen*, Yun Tang*
期刊: Euro. J. Med. Chem.
信息: 2011 | Vol.46 | 4212-4218

2010

6
2010
Triazole-linked benzylated glucosyl, galacotosyl and mannosyl monomers and dimmers as novel sugar scaffold-based PTP1B inhibitors
作者: Zhang Yinjie, He Xiaopeng, Li Cui, Li Zhen, Shi Detai, Gao Lixin, Qiu Beiying, Shi Xiaoxin, Tang Yun*, Li Jia*, Chen Guorong*
期刊: Chem. Lett.
信息: 2010 | 39(12) | 1261-1263
2010
Pharmacophore modeling of human adenosine receptor A2A antagonists
作者: Zhejun Xu, Feixiong Cheng, Chenxiao Da, Guixia Liu and Yun Tang*
期刊: J. Mol .Model
信息: 2010 | Vol.16 | 1867-1876
2010
Insights into binding modes of adenosine A2B antagonists with ligand-based and receptor-based methods
作者: Feixiong Cheng, Zhejun Xu, Liu Guixia and Yun Tang*
期刊: Euro. J. Med. Chem.
信息: 2010 | Vol.45 | 3459-3471
2010
Accuracy Assessment of Protein-Based Docking Programs against RNA Targets
作者: Yaozong Li, Jie Shen, Xianqiang Sun, Weihua Li, Guixia Liu, and Yun Tang*
期刊: J. Chem. Inf. Model
信息: 2010 | Vol.50 | 1134-146
2010
Estimation of ADME Properties with Substructure Pattern Recognition
作者: Jie Shen, Feixiong Cheng, You Xu, Weihua Li,* and Yun Tang*
期刊: J. Chem. Inf. Model.
信息: 2010 | Vol.50 | 1034-041
2010
Discovery of Potent Ligands for Estrogen Receptor β by Structure-Based Virtual Screening
作者: Jie Shen, Chengfang Tan, Yanyan Zhang, Xi Li, Weihua Li, Jin Huang,,Xu Shen and Yun Tang
期刊: J. Med. Chem.
信息: 2010 | Vol.53 | 5361-365

2009

4
2009
The crystal structure of a complex of acetylcholinesterase with a bis-(-)-nor-meptazinol derivative reveals disruption of the catalytic triad
作者: Paz A, Xie Q, Greenblatt HM, Fu W, Tang Y, Silman I, Qiu ZB, Sussman JL*
期刊: J. Med. Chem.
信息: 2009 | 52(8) | 2543-2549
2009
Reduced catalytic activity of P450 2A6 mutants with Coumarin: a computational investigation
作者: Li WH, Ode H, Hoshino T*, Liu H, Tang Y*, Jiang HL
期刊: J. Chem. Theory Comput.
信息: 2009 | 5(5) | 1411-1420
2009
Computational Insights into the Mechanism of Ligand Unbinding and Selectivity of Estrogen Receptors
作者: Jie Shen, Weihua Li, Guixia Liu, Yun Tang and Hualiang Jiang
期刊: J. Phys. Chem. B
信息: 2009 | 113(30) | 10436-0444
2009
Structure–function analysis of human protein Ero1-La
作者: Yanyan Chu, Charles Yang, Xianjun Chen, Wenyun Zheng, Yi Yang* and Yun Tang,*
期刊: Biochem. Biophys. Res. Comm.
信息: 2009 | Vol.389 | 645-650

2008

7
2008
Hyrtiosal, from the marine sponge Hyrtios erectus, inhibits HIV-1 integrase binding to viral DNA by a new inhibitor binding site
作者: Du L, Shen LL, Yu ZG, Chen J, Guo YW*, Tang Y*, Shen X*, Jiang HL
期刊: ChemMedChem
信息: 2008 | 3(1) | 173-180
2008
Insights into ligand selectivity in estrogen receptor isoforms: molecular dynamics simulations and binding free energy calculations
作者: Zeng J, Li WH, Zhao YX, Liu GX*, Tang Y*, Jiang HL
期刊: J. Phys. Chem. B
信息: 2008 | 112(9) | 2719-2726
2008
Probing ligand binding modes of human cytochrome P450 2J2 by homology modeling, molecular dynamics simulation, and flexible molecular docking
作者: Li WH, Tang Y*, Liu H, Cheng JG, Zhu WL, Jiang HL
期刊: Proteins
信息: 2008 | 71(2) | 938-949
2008
Insights into the interactions between HIV-1 integrase and human LEDGF/p75 by molecular dynamics simulation and free energy calculation
作者: Zhao YX, Li WH, Zeng J, Liu GX, Tang Y*
期刊: Proteins
信息: 2008 | 72(2) | 635-645
2008
In silico prediction of blood-brain partitioning using a chemometric method called genetic algorithm based variable selection
作者: Shen J, Du YP, Zhao YX, Liu GX, Tang Y*
期刊: QSAR Comb. Sci.
信息: 2008 | 27(6) | 704-717
2008
Role of acetylation and extra-cellular location of heat shock protein 90alpha in tumor cell invasion
作者: Yang YH, Rao R, Shen J, Tang Y, Fiskus W, Nechtman J, Atadja P, Bhalla K
期刊: Cancer Res.
信息: 2008 | 68(12) | 4833-4842
2008
D77, one benzoic acid derivative, functions as a novel anti-HIV-1 inhibitor targeting the interaction between integrase and cellular LEDGF/p75
作者: Du L, Zhao YX, Chen J, Yang LM, Zheng YT, Tang Y*, Shen X*, Jiang HL
期刊: Biochem. Biophys. Res. Comm.
信息: 2008 | 375(1) | 139-144

2007

2
2007
Synthesis of highly functionalized chiral cyclopentanes by catalytic enantio- and diastereoselective double Michael addition reactions
作者: Zu L, Li H, Xie H, Wang J, Jiang W, Tang Y*, Wang W*
期刊: Angew. Chem. Int. Ed.
信息: 2007 | 46(20) | 3732-3734
2007
Structure-based 3D-QSAR studies on heteroarylpiperazine derivatives as 5-HT3 receptor antagonists
作者: Zhou YJ, Zhu LP, Tang Y*, Ye DY*
期刊: Eur. J. Med. Chem.
信息: 2007 | 42(7) | 977-984

2006

4
2006
Molecular modeling and 3D-QSAR studies of indolomorphinan derivatives as kappa opioid antagonists
作者: Li W, Tang Y*, Zheng YL, Qiu ZB*
期刊: Bioorg. Med. Chem.
信息: 2006 | 14(3) | 601-610
2006
QSAR study of 4-phenylpiperidine derivatives as mu opioid agonists by neural network method
作者: Wang XH, Tang Y*, Xie Q, Qiu ZB*
期刊: Eur. J. Med. Chem.
信息: 2006 | 41(2) | 226-232
2006
Action mechanisms and structure–activity relationships of PI3Kγ inhibitors on the enzyme: a molecular modeling study
作者: Kuang RR, Qian F, Li Z, Wei DZ*, Tang Y*
期刊: Eur. J. Med. Chem.
信息: 2006 | 41(4) | 558-565
2006
New technologies of computer-aided drug design: towards target identification and new chemical entity discovery
作者: Tang Y, Zhu WL, Chen KX, Jiang HL*
期刊: Drug Disc. Today: Technologies
信息: 2006 | 3(3) | 307-313